SCHEMBL16004231

SCHEMBL16004231

Cc1ccc(S(=O)(=O)N2CCOc3ccc(COCc4cccc(F)c4)cc3C2)cc1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PKM P14618 7/20 0.53
ALDH1A1 P00352 5/20 0.53
PKLR P30613 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
LMNA P02545 6/20 0.42
TSHR P16473 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
SMN1; SMN2 Q16637 4/20 0.41
MAPT P10636 2/20 0.41
TP53 P04637 1/20 0.41
POLB P06746 2/20 0.41
RORC P51449 1/20 0.40
CRHBP P24387 1/20 0.40
CRHR2 Q13324 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16004230 0.92 PKM (0.46) PKMALDH1A1PKLRLMNANPSR1
SCHEMBL16004017 0.91 PKM (0.44) PKMALDH1A1PKLRLMNASMN1; SMN2
SCHEMBL16004333 0.90 PKM (0.47) PKMALDH1A1PKLRLMNANPSR1
SCHEMBL16004331 0.88 PKM (0.47) PKMALDH1A1PKLRNPSR1SMN1; SMN2
SCHEMBL16004336 0.86 PKM (0.52) PKMALDH1A1PKLRMEN1KMT2A
SCHEMBL16004327 0.86 PKM (0.51) PKMALDH1A1PKLRMEN1KMT2A
SCHEMBL16004012 0.84 NPC1 (0.41) PKMALDH1A1PKLRMEN1KMT2A
SCHEMBL16004018 0.83 NTRK1 (0.39) PKMALDH1A1PKLR
SCHEMBL16004255 0.81 L3MBTL1 (0.44) PKMPKLRMEN1KMT2ALMNA
SCHEMBL16004016 0.81 PKM (0.43) PKMALDH1A1PKLRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed