SCHEMBL16004336

SCHEMBL16004336

COc1cccc(S(=O)(=O)N2CCOc3ccc(COCc4cccc(F)c4)cc3C2)c1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PKM P14618 8/20 0.52
PKLR P30613 3/20 0.52
POLB P06746 3/20 0.48
MAPT P10636 3/20 0.44
ALDH1A1 P00352 4/20 0.42
MAPK1 P28482 2/20 0.42
LMNA P02545 1/20 0.42
TSHR P16473 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16004230 0.89 PKM (0.46) PKMPKLRALDH1A1MAPK1LMNA
SCHEMBL16004163 0.89 PKM (0.49) PKMPKLRPOLBMAPTALDH1A1
SCHEMBL16004333 0.87 PKM (0.47) PKMPKLRALDH1A1MAPK1LMNA
SCHEMBL16004231 0.86 PKM (0.53) PKMPKLRPOLBMAPTALDH1A1
SCHEMBL16004099 0.85 PKM (0.52) PKMPKLRPOLBMAPTALDH1A1
SCHEMBL16004017 0.85 PKM (0.44) PKMPKLRPOLBALDH1A1MAPK1
SCHEMBL16004331 0.82 PKM (0.47) PKMPKLRPOLBMAPTALDH1A1
SCHEMBL16004012 0.82 NPC1 (0.41) PKMPKLRPOLBALDH1A1MAPK1
SCHEMBL16004261 0.81 LMNA (0.48) POLBMAPTALDH1A1MAPK1LMNA
SCHEMBL16004327 0.80 PKM (0.51) PKMPKLRPOLBALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed