SCHEMBL16004286

SCHEMBL16004286

CC(=O)N(CCc1ccccc1)Cc1ccc2c(c1)CN(C(=O)NC(C)(C)C)CCO2

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GPR142 Q7Z601 4/20 0.41
ALDH1A1 P00352 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
RIPK1 Q13546 3/20 0.39
CREBBP Q92793 4/20 0.38
FAAH O00519 1/20 0.37
MGLL Q99685 2/20 0.37
NAMPT P43490 3/20 0.37
PIK3CA P42336 1/20 0.37
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16004290 0.90 CREBBP (0.47) GPR142CREBBP
SCHEMBL16004244 0.85 GPR142 (0.37) GPR142ALDH1A1SMN1; SMN2RIPK1CREBBP
SCHEMBL16004117 0.85 KDM4E (0.43) GPR142ALDH1A1SMN1; SMN2RIPK1FAAH
SCHEMBL16004421 0.81 GPR142 (0.43) GPR142ALDH1A1SMN1; SMN2NPSR1
SCHEMBL16004291 0.79 MAPT (0.47) GPR142RIPK1CREBBPNAMPT
SCHEMBL16004068 0.76 MAPT (0.49) GPR142ALDH1A1CREBBPNAMPT
SCHEMBL16003971 0.75 MAPT (0.35) ALDH1A1MGLLNPSR1
SCHEMBL16003966 0.75 MEN1 (0.36) ALDH1A1MGLLNPSR1
SCHEMBL16004278 0.75 GPR142 (0.59) GPR142SMN1; SMN2FAAHNAMPT
SCHEMBL16003967 0.75 LMNA (0.40) ALDH1A1RIPK1MGLLNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed