SCHEMBL16004117

SCHEMBL16004117

CC(=O)N(CCc1ccccc1)Cc1ccc2c(c1)CN(C(=O)CN(C)C)CCO2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.43
LIPG Q9Y5X9 1/20 0.42
ALOX15 P16050 1/20 0.42
CASP1 P29466 1/20 0.42
HSD17B10 Q99714 1/20 0.42
LMNA P02545 2/20 0.40
HTT P42858 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MGLL Q99685 2/20 0.38
KMT2A Q03164 2/20 0.38
GPR142 Q7Z601 2/20 0.38
CHRM5 P08912 1/20 0.38
CHRM1 P11229 1/20 0.38
ALDH1A1 P00352 2/20 0.37
MEN1 O00255 1/20 0.37
MAPT P10636 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
RIPK1 Q13546 2/20 0.37
NAAA Q02083 2/20 0.37
PIK3CA P42336 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16004244 0.89 GPR142 (0.37) KDM4EALOX15CASP1HSD17B10LMNA
SCHEMBL16004290 0.87 CREBBP (0.47) GPR142
SCHEMBL16004236 0.85 KDM4E (0.43) KDM4ESMN1; SMN2KMT2AGPR142ALDH1A1
SCHEMBL16004286 0.85 GPR142 (0.41) SMN1; SMN2MGLLGPR142ALDH1A1NPSR1
SCHEMBL16004233 0.81 GPR142 (0.47) LMNASMN1; SMN2KMT2AGPR142ALDH1A1
SCHEMBL16004421 0.79 GPR142 (0.43) KDM4EHSD17B10LMNASMN1; SMN2KMT2A
SCHEMBL16003966 0.77 MEN1 (0.36) KDM4ELMNAHTTMGLLKMT2A
SCHEMBL16003971 0.77 MAPT (0.35) KDM4ELMNAHTTMGLLKMT2A
SCHEMBL16003967 0.77 LMNA (0.40) KDM4ELMNAHTTMGLLKMT2A
SCHEMBL16003968 0.77 ALDH1A1 (0.42) KDM4ELMNAHTTMGLLKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed