SCHEMBL16023924

SCHEMBL16023924

COc1ccc(Cn2nc(N(C)C)nc2Nc2cc(Cl)cc(Cl)c2)cc1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 5/20 0.41
NPBWR1 P48145 6/20 0.39
SMN1; SMN2 Q16637 2/20 0.37
KDR P35968 1/20 0.37
P2RX3 P56373 2/20 0.37
PDE10A Q9Y233 1/20 0.37
MCHR1 Q99705 1/20 0.36
BUB1 O43683 1/20 0.36
CXCR2 P25025 1/20 0.36
MEN1 O00255 1/20 0.36
HTT P42858 1/20 0.36
KMT2A Q03164 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16023925 0.88 NPBWR1 (0.40) P2RX7NPBWR1P2RX3PDE10AMCHR1
SCHEMBL16014856 0.86 P2RX7 (0.44) P2RX7NPBWR1SMN1; SMN2KDRP2RX3
SCHEMBL16014805 0.85 P2RX7 (0.43) P2RX7NPBWR1KDRP2RX3MCHR1
SCHEMBL16014593 0.84 P2RX7 (0.42) P2RX7NPBWR1KDRP2RX3MCHR1
SCHEMBL16014705 0.84 P2RX7 (0.47) P2RX7NPBWR1P2RX3BUB1MEN1
SCHEMBL16014562 0.82 P2RX7 (0.41) P2RX7NPBWR1KDRP2RX3PDE10A
SCHEMBL16014715 0.80 P2RX7 (0.42) P2RX7NPBWR1P2RX3MCHR1
SCHEMBL16023894 0.77 SMN1; SMN2 (0.38) P2RX7NPBWR1SMN1; SMN2PDE10A
SCHEMBL16014359 0.75 P2RX7 (0.41) P2RX7NPBWR1SMN1; SMN2KDRP2RX3
SCHEMBL16014845 0.74 ALDH1A1 (0.41) NPBWR1SMN1; SMN2MEN1HTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014135472-A1 ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2014-09-12 WO disclosed