SCHEMBL16023925

SCHEMBL16023925

COc1ccc(Cn2nc(N(C)C)nc2Nc2cc(Cl)c(Br)c(Cl)c2)cc1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NPBWR1 P48145 10/20 0.40
P2RX7 Q99572 2/20 0.38
P2RX3 P56373 2/20 0.37
MCHR1 Q99705 1/20 0.36
DCTPP1 Q9H773 1/20 0.36
HTT P42858 1/20 0.36
PDE10A Q9Y233 1/20 0.35
BUB1 O43683 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16023924 0.88 P2RX7 (0.41) NPBWR1P2RX7P2RX3MCHR1HTT
SCHEMBL16014642 0.86 NPBWR1 (0.42) NPBWR1P2RX7P2RX3MCHR1DCTPP1
SCHEMBL16014737 0.81 NPBWR1 (0.41) NPBWR1P2RX7P2RX3MCHR1
SCHEMBL16014625 0.78 P2RX7 (0.48) NPBWR1P2RX7MCHR1
SCHEMBL16014593 0.77 P2RX7 (0.42) NPBWR1P2RX7P2RX3MCHR1DCTPP1
SCHEMBL16014845 0.76 ALDH1A1 (0.41) NPBWR1HTT
SCHEMBL16014856 0.74 P2RX7 (0.44) NPBWR1P2RX7P2RX3MCHR1DCTPP1
SCHEMBL16014805 0.73 P2RX7 (0.43) NPBWR1P2RX7P2RX3MCHR1DCTPP1
SCHEMBL16014359 0.73 P2RX7 (0.41) NPBWR1P2RX7P2RX3MCHR1DCTPP1
SCHEMBL16014705 0.72 P2RX7 (0.47) NPBWR1P2RX7P2RX3BUB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014135472-A1 ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2014-09-12 WO disclosed