SCHEMBL16066906

SCHEMBL16066906

CCCCOc1ccc(C(=O)C(O)O)c2ccc(=O)[nH]c12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 5/20 0.42
CNR1 P21554 4/20 0.42
CYP2C9 P11712 1/20 0.39
ALDH1A1 P00352 3/20 0.36
TSHR P16473 2/20 0.36
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
LMNA P02545 2/20 0.36
MAPT P10636 2/20 0.36
NR1I2 O75469 1/20 0.36
CHRM2 P08172 1/20 0.36
CYP3A4 P08684 1/20 0.36
ADRA2A P08913 1/20 0.36
OPRK1 P41145 1/20 0.36
HTR2B P41595 1/20 0.36
SLC6A3 Q01959 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
ADRB2 P07550 1/20 0.35
CA9 Q16790 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13618088 0.86 CA9 (0.42) CNR2CNR1CYP2C9ALDH1A1TSHR
SCHEMBL13589496 0.85 CNR2 (0.41) CNR2CNR1CYP2C9ALDH1A1TSHR
SCHEMBL16066899 0.83 CNR2 (0.39) CNR2CNR1CYP2C9ALDH1A1TSHR
SCHEMBL13617611 0.83 HPGDS (0.42) CNR2CNR1CYP2C9ALDH1A1TSHR
SCHEMBL30862093 0.82 KDM4E (0.42) ALDH1A1TSHRKDM4EMEN1KMT2A
SCHEMBL2798225 0.81 MMP1 (0.41) ALDH1A1MEN1KMT2AMAPTADRB2
SCHEMBL1205431 0.80 SMN1; SMN2 (0.41) CNR2CNR1CYP2C9ALDH1A1MEN1
SCHEMBL13617868 0.79 ADRB2 (0.47) CYP2C9TSHRKDM4EMEN1KMT2A
SCHEMBL15630202 0.78 ADRB2 (0.43) CYP2C9TSHRKDM4EMEN1KMT2A
SCHEMBL13617663 0.78 ADRB2 (0.44) CYP2C9TSHRKDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014139485-A1 A METHOD FOR THE PREPARATION OF 5-[(R)-2-(5,6-DIETHYL-INDAN-2-YLAMINO)-L-HYDROXYETHYL]- 8-HYDROXY-(1H)-QUINOLIN-2-ONE (INDACATEROL) ZENTIVA, K.S. (CZ) 2014-09-18 WO disclosed