SCHEMBL16099686

SCHEMBL16099686

Oc1cc(C(F)(F)F)c2c3ccncc3n(CCN3CCOCC3)c2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFATC1 O95644 1/20 0.41
GSK3B P49841 1/20 0.41
DYRK1A Q13627 1/20 0.41
CHEK1 O14757 3/20 0.36
WEE1 P30291 3/20 0.36
CYP1A2 P05177 3/20 0.36
CYP2D6 P10635 3/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2C19 P33261 2/20 0.36
HIF1A Q16665 2/20 0.36
LMNA P02545 1/20 0.36
CDK1 P06493 1/20 0.35
CCNB1 P14635 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.34
ALOX15 P16050 2/20 0.34
GAA P10253 1/20 0.34
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16099658 0.84 NFATC1 (0.43) NFATC1GSK3BDYRK1ACHEK1WEE1
SCHEMBL16100179 0.81 PLK1 (0.43) CNR2
SCHEMBL16098852 0.81 HASPIN (0.45) NFATC1GSK3BDYRK1ALMNAGAA
SCHEMBL16097995 0.80 CYP2D6 (0.38) DYRK1ACHEK1WEE1CYP2D6CNR2
SCHEMBL2565027 0.80 HASPIN (0.49) CYP1A2CYP2D6CYP3A4HIF1AALOX15
SCHEMBL16093943 0.79 NFATC1 (0.47) NFATC1GSK3BDYRK1ACHEK1WEE1
SCHEMBL16099365 0.76 CYP2D6 (0.35) CYP2D6KDM4EHSD17B10ALDH1A1MAPK13
SCHEMBL25499004 0.75 NFATC1 (0.43) NFATC1GSK3BDYRK1ACYP1A2CYP2D6
SCHEMBL21711353 0.72 NFATC1 (0.43) NFATC1GSK3BDYRK1ACYP1A2CYP2D6
SCHEMBL16099754 0.72 HASPIN (0.45) NFATC1GSK3BDYRK1ACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2968284-A2 ALKYL-AMINE HARMINE DERIVATIVES FOR PROMOTING BONE GROWTH Osteoqc Inc. (CA) 2016-01-20 EP disclosed
WO-2014153203-A2 ALKYL-AMINE HARMINE DERIVATIVES FOR PROMOTING BONE GROWTH OSSIFI INC. (US) 2014-09-25 WO disclosed