SCHEMBL16100969

SCHEMBL16100969

Cc1cccc(N=CCc2cnn(C)c2)c1O[SiH](C)C

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.32
GABRA5 P31644 1/20 0.32
KCNH2 Q12809 2/20 0.31
JAK2 O60674 1/20 0.31
JAK1 P23458 1/20 0.31
TYK2 P29597 1/20 0.31
JAK3 P52333 1/20 0.31
PDCD1LG2 Q9BQ51 1/20 0.30
CD274 Q9NZQ7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16101361 0.87 PDCD1LG2 (0.35) KCNH2JAK2JAK1TYK2JAK3
SCHEMBL16101324 0.85 JAK2 (0.31) JAK2JAK1TYK2JAK3PDCD1LG2
SCHEMBL16101394 0.84 GABRA1 (0.32) GABRA1GABRA5JAK2JAK1TYK2
SCHEMBL17499285 0.83 GABRA1 (0.35) GABRA1GABRA5
SCHEMBL28823574 0.83 GABRA1 (0.31) GABRA1GABRA5JAK2JAK1TYK2
SCHEMBL28039892 0.79 KDM4E (0.31)
SCHEMBL16102408 0.78 HPGD (0.31)
SCHEMBL16101151 0.78 HPGD (0.31)
SCHEMBL28039907 0.77 HPGD (0.30)
SCHEMBL28039879 0.77 HPGD (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2969593-B1 POLYMERS FUNCTIONALIZED WITH HETEROCYCLIC IMINES BRIDGESTONE CORP (JP) 2020-11-04 EP disclosed
US-9850328-B2 Polymers functionalized with heterocyclic imines BRIDGESTONE CORPORATION (JP) 2017-12-26 US disclosed
US-20160039958-A1 Polymers Functionalized With Heterocyclic Imines BRIDGESTONE CORPORATION (JP) 2016-02-11 US disclosed
EP-2969593-A1 POLYMERS FUNCTIONALIZED WITH HETEROCYCLIC IMINES Bridgestone Corporation (JP) 2016-01-20 EP disclosed
WO-2014149931-A1 POLYMERS FUNCTIONALIZED WITH HETEROCYCLIC IMINES BRIDGESTONE CORPORATION (JP) 2014-09-25 WO disclosed