SCHEMBL16112307

SCHEMBL16112307

O=C(c1cc(-c2ccccc2Cl)c[nH]1)N(O)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNC P24863 1/20 0.41
CDK8 P49336 1/20 0.41
ALDH1A1 P00352 2/20 0.40
MAPK1 P28482 4/20 0.40
NOTUM Q6P988 1/20 0.39
ALPL P05186 1/20 0.39
CYP2A6 P11509 1/20 0.39
IKBKB O14920 1/20 0.37
PDK1 Q15118 1/20 0.37
POLB P06746 2/20 0.36
GPBAR1 Q8TDU6 1/20 0.35
KAT6A Q92794 1/20 0.35
KDM4E B2RXH2 1/20 0.35
HPGD P15428 1/20 0.35
MTNR1A P48039 1/20 0.35
MTNR1B P49286 1/20 0.35
PRKAB2 O43741 1/20 0.35
PRKAG1 P54619 1/20 0.35
PRKAA2 P54646 1/20 0.35
PRKAA1 Q13131 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16112230 0.84 MAPK1 (0.43) CCNCCDK8ALDH1A1MAPK1NOTUM
SCHEMBL1990297 0.70 GABRP (0.52) CCNCCDK8ALDH1A1MAPK1ALPL
SCHEMBL16112306 0.69 DOT1L (0.41) CCNCCDK8ALDH1A1MAPK1NOTUM
SCHEMBL10901104 0.69 DYRK1A (0.58) ALDH1A1ALPLCYP2A6IKBKBKDM4E
SCHEMBL16111746 0.69 GAA (0.46) CCNCCDK8ALDH1A1ALPLMEN1
SCHEMBL5924860 0.68 CYP2A6 (0.54) ALDH1A1ALPLCYP2A6IKBKBKAT6A
SCHEMBL15124553 0.68 CYP2A6 (0.54) ALDH1A1ALPLCYP2A6IKBKBKAT6A
SCHEMBL11265372 0.66 POLB (0.46) ALDH1A1POLBGPBAR1KDM4EHPGD
SCHEMBL5820946 0.66 TSHR (0.44) KDM4EHPGD
SCHEMBL16117898 0.66 JAK3 (0.43) ALDH1A1MAPK1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014159214-A1 HISTONE DEACETYLASE INHIBITORS AND COMPOSITIONS AND METHODS OF USE THEREOF CHDI FOUNDATION, INC. (US) 2014-10-02 WO disclosed