SCHEMBL16112306

SCHEMBL16112306

O=C(NO)c1cc(-c2ccccc2-c2ccccc2Cl)c[nH]1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DOT1L Q8TEK3 1/20 0.41
CCNC P24863 2/20 0.40
CDK8 P49336 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
HDAC8 Q9BY41 2/20 0.39
MAPK14 Q16539 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
MAPK1 P28482 3/20 0.39
NOTUM Q6P988 1/20 0.38
ALPL P05186 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
MAPK10 P53779 1/20 0.36
KAT6A Q92794 1/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16112229 0.83 CCNC (0.40) CCNCCDK8HDAC8MAPK14MEN1
SCHEMBL16111746 0.82 GAA (0.46) CCNCCDK8MAPK14ALPLMEN1
SCHEMBL20792373 0.77 MAPK14 (0.62) MAPK14MEN1KMT2AALDH1A1
SCHEMBL20792417 0.72 HSD11B1 (0.46) CCNCCDK8MAPK14MEN1KMT2A
SCHEMBL20792371 0.72 HTT (0.56) ALDH1A1
SCHEMBL1990297 0.69 GABRP (0.52) CCNCCDK8MAPK1ALPLMEN1
SCHEMBL16112307 0.69 CCNC (0.41) CCNCCDK8MAPK1NOTUMALPL
SCHEMBL20792432 0.68 MAPK14 (0.40) CCNCCDK8MAPK14MAPK1MEN1
SCHEMBL5944029 0.67 HDAC6 (0.61) HDAC6HDAC8HDAC3HDAC1HDAC2
SCHEMBL16112586 0.66 ALDH1A1 (0.46) CCNCCDK8ALPLMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014159214-A1 HISTONE DEACETYLASE INHIBITORS AND COMPOSITIONS AND METHODS OF USE THEREOF CHDI FOUNDATION, INC. (US) 2014-10-02 WO disclosed