SCHEMBL16112355

SCHEMBL16112355

Clc1ccc(Br)cc1-c1nccs1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
HTT P42858 1/20 0.39
PDPK1 O15530 1/20 0.39
ABL1 P00519 1/20 0.38
BCR P11274 1/20 0.38
FBP1 P09467 2/20 0.37
ADORA2A P29274 2/20 0.37
ADORA1 P30542 1/20 0.37
THRA P10827 1/20 0.36
THRB P10828 1/20 0.36
CYP1A1 P04798 2/20 0.35
CYP1A2 P05177 2/20 0.35
CYP1B1 Q16678 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2029417 0.82 FBP1 (0.45) MAPTKDM4EMEN1NPC1ALDH1A1
SCHEMBL2653159 0.79 PDPK1 (0.39) MEN1NPC1RAB9AKMT2APDPK1
SCHEMBL2902222 0.76 F2RL1 (0.40) MEN1NPC1RAB9AKMT2APDPK1
SCHEMBL11440352 0.76 ADORA2A (0.41) ALDH1A1PDPK1ABL1BCRFBP1
SCHEMBL4047151 0.76 PDPK1 (0.39) MEN1NPC1RAB9AKMT2APDPK1
SCHEMBL16990890 0.76 PDPK1 (0.56) NPC1RAB9APDPK1ABL1BCR
SCHEMBL16112533 0.74 ADRA1A (0.40) PDPK1ABL1BCRFBP1ADORA2A
SCHEMBL1565328 0.74 PDPK1 (0.53) MAPTKDM4EMEN1NPC1ALDH1A1
SCHEMBL30457805 0.74 PDPK1 (0.53) MAPTKDM4EMEN1NPC1ALDH1A1
SCHEMBL27468615 0.73 HSD17B10 (0.49) MAPTKDM4EMEN1NPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2968233-A1 HISTONE DEACETYLASE INHIBITORS AND COMPOSITIONS AND METHODS OF USE THEREOF CHDI Foundation, Inc. (US) 2016-01-20 EP disclosed
WO-2014159224-A1 HISTONE DEACETYLASE INHIBITORS AND COMPOSITIONS AND METHODS OF USE THEREOF CHDI FOUNDATION, INC. (US) 2014-10-02 WO disclosed