SCHEMBL16136391

SCHEMBL16136391

CC(C)(C)[SiH](OCCc1ccc(CBr)cc1)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TSHR P16473 1/20 0.38
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
PPARG P37231 5/20 0.33
PPARA Q07869 3/20 0.33
TDP1 Q9NUW8 1/20 0.32
PPARD Q03181 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16136456 0.91 IDO1 (0.37) TRPA1ALDH1A1TSHRCES2CES1
SCHEMBL27538454 0.89 CA1 (0.37) ALDH1A1CES1PPARGPPARATDP1
SCHEMBL705121 0.75 MEN1 (0.35) ALDH1A1TSHR
SCHEMBL707593 0.72 LTA4H (0.42) ALDH1A1TSHRTDP1
SCHEMBL713132 0.71 RELA (0.33) ALDH1A1TSHR
SCHEMBL28519614 0.71 TRPA1 (0.36) TRPA1ALDH1A1TSHRCES2CES1
SCHEMBL703504 0.70 CA1 (0.40) ALDH1A1TDP1
SCHEMBL3681371 0.67 TRPA1 (0.38) TRPA1ALDH1A1TSHRCES2CES1
SCHEMBL10516808 0.66 MAPK1 (0.37) ALDH1A1
SCHEMBL27884138 0.66 NPC1 (0.56) TRPA1ALDH1A1TSHRPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1813611-B1 1-SUBSTITUTED-3- BETA-D-GLYCOPYRANOSYLATED NITROGENOUS HETERO- CYCLIC COMPOUNDS AND MEDICINES CONTAINING THE SAME KISSEI PHARMACEUTICAL (JP) 2014-10-01 EP disclosed