SCHEMBL16136559

SCHEMBL16136559

CC1c2ccc(-c3cccc(C#N)c3)cc2C(=O)CC1c1cccnc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 2/20 0.42
CYP11B2 P19099 3/20 0.41
CYP11B1 P15538 2/20 0.41
CYP17A1 P05093 1/20 0.41
STK10 O94804 2/20 0.41
SLK Q9H2G2 2/20 0.41
NEK1 Q96PY6 1/20 0.40
DGAT2 Q96PD7 1/20 0.40
FLT3 P36888 2/20 0.40
CHRNB2 P17787 1/20 0.39
CHRNA5 P30532 1/20 0.39
CHRNA4 P43681 1/20 0.39
KDM1A O60341 1/20 0.39
CREBBP Q92793 1/20 0.38
SLC22A12 Q96S37 1/20 0.37
F2R P25116 1/20 0.37
ALDH1A1 P00352 2/20 0.37
CYP1A2 P05177 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2C19 P33261 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1821928 0.77 CYP19A1 (0.47) PGRCYP11B2CYP11B1CYP17A1STK10
SCHEMBL29809001 0.69 CYP11B2 (0.71) CYP11B2CYP11B1CYP17A1NEK1CHRNB2
SCHEMBL13537172 0.69 CYP11B2 (0.71) CYP11B2CYP11B1CYP17A1NEK1CHRNB2
SCHEMBL2376622 0.68 CHRNB2 (0.39) CYP11B2CYP11B1CYP17A1NEK1FLT3
SCHEMBL2376620 0.68 CHRNB2 (0.39) CYP11B2CYP11B1CYP17A1NEK1FLT3
SCHEMBL3921199 0.63 MAOB (0.51) PGRKDM1ACREBBPCLK4
SCHEMBL1822896 0.62 CYP19A1 (0.44) PGRCYP3A4CLK4
SCHEMBL13297269 0.62 PGR (0.48) PGRCREBBPSLC22A12CLK4
SCHEMBL1805616 0.62 CHEK1 (0.44) PGRCHRNB2CHRNA4CREBBPSLC22A12
SCHEMBL1805619 0.62 CHEK1 (0.44) PGRCHRNB2CHRNA4CREBBPSLC22A12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2324032-B1 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS INC (US) 2014-10-01 EP disclosed