SCHEMBL29809001

SCHEMBL29809001

N#Cc1cccc(-c2cccnc2)c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 4/20 0.71
CYP11B1 P15538 3/20 0.71
CYP17A1 P05093 1/20 0.71
CHRNB2 P17787 2/20 0.64
CHRNA5 P30532 2/20 0.64
CHRNA4 P43681 2/20 0.64
NEK1 Q96PY6 1/20 0.59
CLK4 Q9HAZ1 4/20 0.58
ALDH1A1 P00352 4/20 0.56
CYP1A2 P05177 4/20 0.56
CYP3A4 P08684 4/20 0.56
CYP2A6 P11509 1/20 0.56
MEN1 O00255 1/20 0.55
PSIP1 O75475 1/20 0.55
AXL P30530 1/20 0.55
MKNK1 Q9BUB5 1/20 0.55
MKNK2 Q9HBH9 1/20 0.55
IDO1 P14902 2/20 0.54
CYP19A1 P11511 1/20 0.54
GABRA1 P14867 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13537172 1.00 CYP11B2 (0.71) CYP11B2CYP11B1CYP17A1CHRNB2CHRNA5
SCHEMBL1690481 0.85 CYP11B2 (0.68) CYP11B2CYP11B1CYP17A1CHRNB2CHRNA5
Benzonitrile SCHEMBL29165371 0.85 CYP11B2 (0.79) CYP11B2CYP11B1CYP17A1CHRNB2CHRNA5
SCHEMBL1422883 0.84 CHRNB2 (0.67) CYP11B2CYP11B1CYP17A1CHRNB2CHRNA5
SCHEMBL18890284 0.83 IDO1 (0.56) CYP11B2CYP11B1CYP17A1CHRNB2CHRNA5
SCHEMBL4511285 0.83 CYP11B2 (1.00) CYP11B2CYP11B1CYP17A1CHRNB2CHRNA5
SCHEMBL3608623 0.82 CHRNB2 (0.54) CYP11B2CYP11B1CYP17A1CHRNB2CHRNA5
SCHEMBL2154026 0.82 CLK4 (0.65) CLK4IDO1GABRA1GABRG2GABRB3
SCHEMBL29984880 0.81 CYP2A6 (0.56) CYP11B2CYP11B1CYP17A1CHRNB2CHRNA5
SCHEMBL28881990 0.81 CYP2A6 (0.56) CYP11B2CYP11B1CYP17A1CHRNB2CHRNA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117567435-A Glutamine cyclase inhibitor and application thereof 上海市第十人民医院 2024-02-20 CN disclosed
CN-114805341-B Aromatic heterocyclic compound, and preparation method and application thereof 上海翊石医药科技有限公司 2023-12-08 CN disclosed
CN-114805341-A Aromatic heterocyclic compounds and preparation method and application thereof 上海翊石医药科技有限公司 2022-07-29 CN disclosed