SCHEMBL16156325

SCHEMBL16156325

COc1c(CBr)ccc2[nH]c(C#N)cc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.36
DRD2 P14416 2/20 0.36
ADRB2 P07550 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
MAPT P10636 2/20 0.33
TSHR P16473 1/20 0.33
GFER P55789 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PTGDR Q13258 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
TUBB4A P04350 1/20 0.30
TUBB P07437 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30406469 0.81 MEN1 (0.36) HTR1ADRD2ADRB2CYP1A2CYP3A4
SCHEMBL25421574 0.81 MEN1 (0.36) HTR1ADRD2ADRB2CYP1A2CYP3A4
SCHEMBL16031335 0.79 STING1 (0.38) HTR1ADRD2ADRB2CYP1A2CYP3A4
SCHEMBL30405780 0.74 ALDH1A1 (0.38) HTR1ADRD2ADRB2CYP1A2CYP3A4
SCHEMBL25421875 0.74 ALDH1A1 (0.38) HTR1ADRD2ADRB2CYP1A2CYP3A4
SCHEMBL19369444 0.73 HTR1A (0.41) HTR1ADRD2ADRB2CYP1A2CYP3A4
SCHEMBL17522629 0.70 PTGDR (0.38) HTR1ADRD2ADRB2CYP1A2CYP3A4
SCHEMBL20259615 0.69 HTR1A (0.38) HTR1ADRD2ADRB2CYP1A2CYP3A4
SCHEMBL20504885 0.68 ADRB2 (0.52) ADRB2CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL28812480 0.68 AOC3 (0.38) CYP1A2KDM4EALDH1A1MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014164543-A1 COMPOSITIONS COMPRISING THIENOPYRIMIDINE AND THIENOPYRIDINE COMPOUNDS AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2014-10-09 WO disclosed