SCHEMBL16181747

SCHEMBL16181747

O=C(NCCI)c1cccnc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.68
MEN1 O00255 5/20 0.66
KMT2A Q03164 5/20 0.66
RAB9A P51151 4/20 0.66
NPC1 O15118 3/20 0.66
SMN1; SMN2 Q16637 3/20 0.66
EPHX2 P34913 4/20 0.62
CYP2C9 P11712 2/20 0.62
CYP2C19 P33261 2/20 0.62
CYP1A2 P05177 1/20 0.62
CYP3A4 P08684 1/20 0.62
MAPT P10636 1/20 0.61
ALDH1A1 P00352 1/20 0.61
GAA P10253 1/20 0.60
ALOX15 P16050 1/20 0.59
HSD17B10 Q99714 1/20 0.59
TDP1 Q9NUW8 1/20 0.59
HDAC1 Q13547 1/20 0.59
HDAC6 Q9UBN7 1/20 0.59
USP2 O75604 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19114989 0.90 EPHX2 (0.68) THRBMEN1KMT2ARAB9ANPC1
SCHEMBL25328235 0.90 THRB (0.77) THRBMEN1KMT2ARAB9ANPC1
SCHEMBL1388180 0.88 THRB (0.70) THRBMEN1KMT2ARAB9ANPC1
SCHEMBL9809561 0.86 RAB9A (0.76) THRBMEN1KMT2ARAB9ANPC1
SCHEMBL17822214 0.86 EPHX2 (0.75) THRBMEN1KMT2ARAB9ANPC1
SCHEMBL3514765 0.85 EPHX2 (0.69) THRBMEN1KMT2ARAB9ANPC1
SCHEMBL30664046 0.85 THRB (0.75) THRBMEN1KMT2ARAB9ANPC1
SCHEMBL5483064 0.85 EPHX2 (0.73) THRBMEN1KMT2ARAB9ANPC1
SCHEMBL62572 0.85 THRB (0.75) THRBMEN1KMT2ARAB9ANPC1
SCHEMBL9763664 0.85 EPHX2 (0.73) THRBMEN1KMT2ARAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017120355-A1 DIHYDROQUINOLINES AND USES THEREOF TEVA PHARMACEUTICAL INDUSTRIES LTD. (IL) 2017-07-13 WO disclosed
EP-2658839-B1 PROCESS FOR THE MANUFACTURE OF NICORANDIL PROCOS SPA (IT) 2014-10-22 EP disclosed