SCHEMBL16190013

SCHEMBL16190013

Fc1c(Br)ccc2c1CCO2

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EED O75530 4/20 0.34
SUZ12 Q15022 4/20 0.34
EZH2 Q15910 4/20 0.34
EGFR P00533 3/20 0.33
MAPT P10636 2/20 0.33
MAOB P27338 1/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
BLM P54132 1/20 0.33
MTNR1B P49286 1/20 0.33
HTR2A P28223 4/20 0.32
HTR2C P28335 4/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
HTR2B P41595 1/20 0.32
KDM1A O60341 2/20 0.32
KCNH2 Q12809 2/20 0.32
KDM1B Q8NB78 2/20 0.32
KIF11 P52732 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31634038 1.00 EED (0.34) EEDSUZ12EZH2EGFRMAPT
SCHEMBL25208990 0.89 HTR2C (0.36) EGFRMAPTMAOBLMNAHTT
SCHEMBL20741822 0.78 HTR2A (0.43) EEDSUZ12EZH2MAPTMAOB
SCHEMBL30949613 0.78 HTR2A (0.43) EEDSUZ12EZH2MAPTMAOB
SCHEMBL30754266 0.76 MTNR1B (0.35) EGFRMAPTMAOBLMNAHTT
SCHEMBL20744138 0.76 HTR2C (0.35) MAPTLMNAHTTBLMMTNR1B
SCHEMBL30684141 0.76 HTR2C (0.35) MAPTLMNAHTTBLMMTNR1B
SCHEMBL1764937 0.76 MTNR1B (0.35) EGFRMAPTMAOBLMNAHTT
SCHEMBL16190012 0.76 HTR2C (0.35) MAPTHTR2AHTR2CHTR2BKIF11
SCHEMBL14720202 0.74 ABCC9 (0.36) MAPTMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025049746-A1 COMPOSITIONS COMPRISING WERNER SYNDROME HELICASE INHIBITORS AND METHODS OF USING THE SAME EIKON THERAPEUTICS, INC. (US) 2025-03-06 WO disclosed
US-12162864-B2 Condensed-cyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2024-12-10 US disclosed
US-20240067668-A1 HETEROARYL DERIVATIVE COMPOUND AND USE THEREOF VORONOI INC. (KR) 2024-02-29 US disclosed
US-20240067668-A1 HETEROARYL DERIVATIVE COMPOUND AND USE THEREOF VORONOI INC. (KR) 2024-02-29 US disclosed
US-20240067668-A1 HETEROARYL DERIVATIVE COMPOUND AND USE THEREOF VORONOI INC. (KR) 2024-02-29 US disclosed
EP-4273149-A1 HETEROARYL DERIVATIVE COMPOUND AND USE THEREOF Voronoi Inc. (KR) 2023-11-08 EP disclosed
US-20230219986-A1 NOVEL AMINOPYRIMIDINE EGFR INHIBITOR QILU PHARMACEUTICAL CO., LTD. (CN) 2023-07-13 US disclosed
US-20230219986-A1 NOVEL AMINOPYRIMIDINE EGFR INHIBITOR QILU PHARMACEUTICAL CO., LTD. (CN) 2023-07-13 US disclosed
EP-4129996-A1 NOVEL AMINOPYRIMIDINE EGFR INHIBITOR QILU PHARMACEUTICAL CO., LTD. (CN) 2023-02-08 EP disclosed
WO-2022146027-A1 HETEROARYL DERIVATIVE COMPOUND AND USE THEREOF 주식회사 비투에스바이오 2022-07-07 WO disclosed
EP-3858823-A1 CONDENSED-CYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2021-08-04 EP disclosed
EP-3858823-A1 CONDENSED-CYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2021-08-04 EP disclosed
WO-2020067457-A1 CONDENSED-CYCLIC COMPOUND 武田薬品工業株式会社 2020-04-02 WO disclosed
WO-2014169845-A2 4,5-DIHYDRO-PYRAZOLO [3, 4-C] PYRID-2-ONES, PREPARATION METHOD AND APPLICATION THEREOF 四川海思科制药有限公司 (CN) 2014-10-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240067668-A1 HETEROARYL DERIVATIVE COMPOUND AND USE THEREOF ERBB2, EGFR, ERBB3 EED 764/4885SUZ12 511/4885EZH2 1494/4885
US-20230219986-A1 NOVEL AMINOPYRIMIDINE EGFR INHIBITOR EGFR, ERBB2, ERBB4 EED 1061/4885SUZ12 1184/4885EZH2 1530/4885
US-12162864-B2 Condensed-cyclic compound SLC10A2, VIP, AVPR2 EED 963/4885SUZ12 653/4885EZH2 597/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.