SCHEMBL16190012

SCHEMBL16190012

Nc1ccc2c(c1F)CCO2

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 8/20 0.35
HTR2A P28223 7/20 0.35
HTR2B P41595 4/20 0.35
DYRK1A Q13627 1/20 0.34
SLC9A1 P19634 4/20 0.33
PRKCI P41743 1/20 0.33
MAPT P10636 2/20 0.32
KDM4E B2RXH2 2/20 0.32
GAA P10253 1/20 0.32
ALDH1A1 P00352 2/20 0.32
SLC9A5 Q14940 1/20 0.31
SLC9A2 Q9UBY0 1/20 0.31
KIF11 P52732 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16190013 0.76 EED (0.34) HTR2CHTR2AHTR2BMAPTKIF11
SCHEMBL31634038 0.76 EED (0.34) HTR2CHTR2AHTR2BMAPTKIF11
SCHEMBL10188136 0.73 MAPT (0.37) MAPTKDM4EGAAALDH1A1
SCHEMBL14203441 0.72 HTR2C (0.36) HTR2CHTR2AHTR2B
SCHEMBL945134 0.71 ITGB2 (0.42) SLC9A1SLC9A5SLC9A2KIF11
SCHEMBL31394265 0.70 LPL (0.35)
Bromide SCHEMBL2483355 0.69 ITGB2 (0.41) SLC9A1SLC9A5SLC9A2KIF11
SCHEMBL25723254 0.69 PKM (0.32) HTR2CHTR2AMAPT
SCHEMBL10818074 0.69 MAPT (0.44) HTR2CHTR2AHTR2BMAPTGAA
SCHEMBL13547884 0.68 HTR2C (0.36) HTR2CHTR2AHTR2BKIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014169845-A2 4,5-DIHYDRO-PYRAZOLO [3, 4-C] PYRID-2-ONES, PREPARATION METHOD AND APPLICATION THEREOF 四川海思科制药有限公司 (CN) 2014-10-23 WO disclosed