SCHEMBL16198239

SCHEMBL16198239

Cc1nccn1-c1ccc(NC(C)C(=O)O)cc1C(F)(F)F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
KDM4E B2RXH2 1/20 0.45
IDH2 P48735 1/20 0.41
NR3C2 P08235 4/20 0.35
CSF1R P07333 2/20 0.35
KIT P10721 2/20 0.35
LYN P07948 1/20 0.35
TEK Q02763 2/20 0.34
RAF1 P04049 1/20 0.34
BRAF P15056 1/20 0.34
MAPK14 Q16539 1/20 0.34
CYP26A1 O43174 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
PORCN Q9H237 1/20 0.34
F2 P00734 1/20 0.34
F10 P00742 1/20 0.34
IDH1 O75874 1/20 0.34
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16198095 0.81 PORCN (0.55) IDH2TEKCYP3A4CYP2D6PORCN
SCHEMBL16198102 0.80 ALDH1A1 (0.45) ALDH1A1KDM4EIDH2NR3C2BRAF
SCHEMBL3528958 0.77 KDM4E (0.51) ALDH1A1KDM4EIDH2NR3C2CSF1R
SCHEMBL16198379 0.77 CYP3A4 (0.49) ALDH1A1NR3C2CYP3A4CYP2D6PORCN
SCHEMBL2467864 0.75 KIT (0.46) KDM4ECSF1RKITLYNTEK
SCHEMBL19951698 0.75 SMN1; SMN2 (0.43) ALDH1A1KDM4ECYP3A4KDR
SCHEMBL1555605 0.75 SMN1; SMN2 (0.43) ALDH1A1KDM4ECYP3A4KDR
SCHEMBL734692 0.73 AR (0.53) ALDH1A1KDM4ECYP3A4
SCHEMBL734816 0.72 KDR (0.59) KDR
SCHEMBL1555612 0.72 KDR (0.59) KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140378429-A1 Carboxamide, Sulfonamide and Amine Compounds and Methods for Using Them RIGEL PHARMACEUTICALS, INC. (US) 2014-12-25 US disclosed
WO-2014175832-A1 WNT PATHWAY MODULATORS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2014-10-30 WO disclosed
WO-2014175832-A1 WNT PATHWAY MODULATORS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2014-10-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140378429-A1 Carboxamide, Sulfonamide and Amine Compounds and Methods for Using Them CPT2, SHMT2, CS ALDH1A1 397/4885KDM4E 3152/4885IDH2 21/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.