SCHEMBL13683096

SCHEMBL13683096

Cn1nc(C(F)(F)F)c(Cl)c1-c1cccnc1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.46
P2RX7 Q99572 3/20 0.45
POLB P06746 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
CYP11B2 P19099 3/20 0.40
ALDH1A1 P00352 3/20 0.39
CYP2A6 P11509 3/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP11B1 P15538 1/20 0.39
MAOA P21397 1/20 0.39
CYP2A13 Q16696 1/20 0.39
NPY5R Q15761 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13430367 0.83 POLB (0.54) LMNAPOLBNPC1RAB9AALDH1A1
SCHEMBL13683098 0.82 KIF11 (0.39) POLBNPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL16200083 0.79 ALDH1A1 (0.48) LMNAP2RX7CYP11B2ALDH1A1CYP2A6
SCHEMBL14039660 0.77 POLB (0.41) LMNAPOLBSMN1; SMN2CYP11B2CYP1A2
SCHEMBL16200054 0.77 P2RX7 (0.45) P2RX7NPC1RAB9ASMN1; SMN2RXFP1
SCHEMBL13066524 0.76 MEN1 (0.46) POLB
SCHEMBL13066522 0.76 SMN1; SMN2 (0.46) LMNAP2RX7POLBSMN1; SMN2
SCHEMBL28851687 0.74 P2RX7 (0.43) LMNAP2RX7NPC1RAB9ASMN1; SMN2
SCHEMBL13682914 0.72 P2RX7 (0.44) LMNAP2RX7POLBNPC1RAB9A
SCHEMBL16200074 0.71 POLB (0.40) LMNAPOLBSMN1; SMN2CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7589199-B2 Substituted piperazines CHEMOCENTRYX, INC. (US) 2009-09-15 US disclosed
US-7435830-B2 Bicyclic and bridged nitrogen heterocycles CHEMOCENTRYX, INC. (US) 2008-10-14 US disclosed