SCHEMBL16200318

SCHEMBL16200318

COc1cc(C)c(C(C)NC(C)=O)cc1Cl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 2/20 0.43
TAS1R3 Q7RTX0 3/20 0.43
TAS1R1 Q7RTX1 3/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MTNR1A P48039 2/20 0.43
MTNR1B P49286 2/20 0.43
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 3/20 0.39
MEN1 O00255 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
LMNA P02545 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
STAT3 P40763 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
RORC P51449 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13683175 0.85 ACACB (0.43) ACACBTAS1R3TAS1R1L3MBTL1MTNR1A
SCHEMBL13683103 0.80 CYP2D6 (0.47) TAS1R3TAS1R1NPC1ALDH1A1
SCHEMBL16200314 0.78 ALDH1A1 (0.38) TAS1R3TAS1R1NPC1RAB9AMEN1
SCHEMBL16200302 0.76 GAA (0.41) L3MBTL1NPC1MEN1KMT2ALMNA
SCHEMBL1754175 0.76 CYP1A2 (0.46) ACACBL3MBTL1SMN1; SMN2MEN1HTT
SCHEMBL16200313 0.76 PGK1 (0.41) TAS1R3TAS1R1NPC1LMNAKDM4E
SCHEMBL2107612 0.74 TNFSF11 (0.46) ACACBTAS1R3TAS1R1L3MBTL1NPC1
SCHEMBL2107613 0.74 TNFSF11 (0.46) ACACBTAS1R3TAS1R1L3MBTL1NPC1
SCHEMBL13178807 0.73 GAA (0.46) NPC1HTTLMNA
SCHEMBL30202757 0.72 GPR139 (0.47) ACACBL3MBTL1NPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720545-B1 BICYCLIC AND BRIDGED NITROGEN HETEROCYCLES CHEMOCENTRYX INC (US) 2014-10-29 EP disclosed