SCHEMBL16215907

SCHEMBL16215907

C=C/C=C\CN1CCCC1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.36
LTA4H P09960 1/20 0.35
HRH3 Q9Y5N1 1/20 0.31
CARM1 Q86X55 1/20 0.31
PRMT6 Q96LA8 1/20 0.31
PRMT8 Q9NR22 1/20 0.31
LMNA P02545 1/20 0.31
CHRNB2 P17787 1/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
CHRNA4 P43681 1/20 0.31
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19720569 1.00 SIGMAR1 (0.36) SIGMAR1LTA4HHRH3CARM1PRMT6
SCHEMBL22972376 0.98 SIGMAR1 (0.38) SIGMAR1LTA4HHRH3CARM1PRMT6
SCHEMBL8520735 0.98 SIGMAR1 (0.38) SIGMAR1LTA4HHRH3CARM1PRMT6
Hydrochloric Acid SCHEMBL2704381 0.95 SIGMAR1 (0.37) SIGMAR1LTA4HHRH3CHRNB2CHRNB4
SCHEMBL9111540 0.78 SIGMAR1 (0.38) SIGMAR1LTA4HHRH3CARM1PRMT6
SCHEMBL9111537 0.78 SIGMAR1 (0.38) SIGMAR1LTA4HHRH3CARM1PRMT6
SCHEMBL23872300 0.78 LTA4H (0.42) SIGMAR1LTA4HHRH3CARM1PRMT6
SCHEMBL819102 0.76 HRH3 (0.37) SIGMAR1HRH3CARM1PRMT6PRMT8
SCHEMBL9112203 0.76 SIGMAR1 (0.41) SIGMAR1LTA4HHRH3CHRNB2CHRNB4
SCHEMBL9112196 0.76 SIGMAR1 (0.41) SIGMAR1LTA4HHRH3CHRNB2CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2470012-B1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME (US) 2014-11-05 EP disclosed