SCHEMBL1622156

SCHEMBL1622156

CC(C)(CNC(=O)C(=O)/C=C/c1ccccc1)c1ccc(F)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAAT5 Q96KN8 6/20 0.50
PLAAT4 Q9UL19 6/20 0.50
PLAAT3 P53816 5/20 0.50
PLAAT2 Q9NWW9 5/20 0.50
LMNA P02545 1/20 0.50
TP53 P04637 1/20 0.50
EGFR P00533 2/20 0.46
MMP1 P03956 1/20 0.46
MMP2 P08253 1/20 0.46
MMP9 P14780 1/20 0.46
CACNA1G O43497 1/20 0.46
CYP1A1 P04798 2/20 0.43
CYP1B1 Q16678 2/20 0.43
MAOB P27338 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
POLB P06746 1/20 0.41
KMT2A Q03164 1/20 0.41
TRPV1 Q8NER1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1620609 0.81 EGFR (0.49) PLAAT5PLAAT4PLAAT3PLAAT2LMNA
SCHEMBL7661577 0.75 PLAAT5 (0.63) PLAAT5PLAAT4PLAAT3PLAAT2LMNA
SCHEMBL12590249 0.75 PLAAT3 (0.47) PLAAT5PLAAT4PLAAT3PLAAT2LMNA
SCHEMBL17240886 0.75 CACNA1G (0.51) LMNATP53CACNA1GSMN1; SMN2NPC1
SCHEMBL6974619 0.73 PLAAT5 (0.65) PLAAT5PLAAT4PLAAT3PLAAT2LMNA
SCHEMBL7660245 0.73 PLAAT5 (0.68) PLAAT5PLAAT4PLAAT3PLAAT2LMNA
SCHEMBL7660641 0.72 PLAAT5 (0.58) PLAAT5PLAAT4PLAAT3PLAAT2LMNA
SCHEMBL6645828 0.71 PLAAT3 (0.57) PLAAT5PLAAT4PLAAT3PLAAT2LMNA
SCHEMBL6977796 0.71 PLAAT5 (0.70) PLAAT5PLAAT4PLAAT3PLAAT2LMNA
SCHEMBL7661326 0.70 PLAAT5 (0.65) PLAAT5PLAAT4PLAAT3PLAAT2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7928134-B2 5-aryl-4,5-dihydro-(1H)-pyrazolines as cannabinoid CB1 receptor agonists SOLVAY PHARMACEUTICALS B.V. (NL) 2011-04-19 US disclosed
US-20090082396-A1 5-ARYL-4,5-DIHYDRO-(1H)-PYRAZOLINES AS CANNABINOID CB1 RECEPTOR AGONISTS SOLVAY PHARMACEUTICALS B.V. 2009-03-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090082396-A1 5-ARYL-4,5-DIHYDRO-(1H)-PYRAZOLINES AS CANNABINOID CB1 RECEPTOR AGONISTS CNR1, CNR2, HTR5A PLAAT5 514/4885PLAAT4 845/4885PLAAT3 1117/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.