SCHEMBL16239076

SCHEMBL16239076

COc1cc(C[C@@H](c2ccccc2)[N+](=O)[O-])ccc1Br

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.40
MAPT P10636 3/20 0.39
HTR2A P28223 2/20 0.39
HPGD P15428 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
KMT2A Q03164 4/20 0.37
MEN1 O00255 2/20 0.37
ALDH1A1 P00352 2/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10474946 0.74 CPA1 (0.47) CYP1A2ALDH1A1
SCHEMBL266009 0.73 MEN1 (0.42) MAPTKMT2AMEN1ALDH1A1
SCHEMBL16239075 0.72 CYP19A1 (0.39) MAPTHPGDCYP1A2KMT2AMEN1
SCHEMBL27653040 0.70 LOXL2 (0.46) ALDH1A1
SCHEMBL2037536 0.70 ALDH1A1 (0.49) LDHAMAPTKMT2AMEN1ALDH1A1
SCHEMBL27968775 0.70 CA2 (0.55) MAPTHTR2AALDH1A1
SCHEMBL27618563 0.68 GABRA1 (0.52) LDHAHTR2ACYP3A4
SCHEMBL27042690 0.68 TAAR1 (0.58) HTR2A
SCHEMBL28046603 0.68 GSR (0.42) MAPTHPGDCYP3A4CYP2D6CYP2C19
SCHEMBL16239369 0.68 ALDH1A1 (0.41) MAPTHPGDCYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8889863-B2 Stereoselective methods, catalysts and intermediates for the synthesis of (−)-Nutlin-3 and related compounds VANDERBILT UNIVERSITY (US) 2014-11-18 US disclosed