SCHEMBL16239491

SCHEMBL16239491

CC1(C)CC(c2ccccc2NS(=O)(=O)c2cccc(F)c2)Nc2c(C(F)(F)F)cccc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC10A2 Q12908 1/20 0.38
SLC10A1 Q14973 1/20 0.38
SLC10A6 Q3KNW5 1/20 0.38
MOGAT2 Q3SYC2 1/20 0.37
KMT2A Q03164 3/20 0.36
DDX3X O00571 2/20 0.36
GAA P10253 2/20 0.36
MEN1 O00255 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
TSHR P16473 1/20 0.34
CYP2C19 P33261 1/20 0.34
SLC22A12 Q96S37 1/20 0.34
PGR P06401 1/20 0.34
JAK1 P23458 1/20 0.34
USP2 O75604 1/20 0.33
POLB P06746 1/20 0.33
LMNA P02545 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16239649 0.92 KMT2A (0.41) KMT2ADDX3XGAAMEN1CYP1A2
SCHEMBL16239499 0.91 KMT2A (0.41) MOGAT2KMT2AGAAMEN1TSHR
SCHEMBL16239852 0.87 SLC10A2 (0.39) SLC10A2SLC10A1SLC10A6KMT2AGAA
SCHEMBL16239817 0.85 SLC22A12 (0.47) KMT2AMEN1CYP1A2CYP3A4CYP2D6
SCHEMBL2137469 0.83 MEN1 (0.40) SLC10A2SLC10A1SLC10A6MOGAT2KMT2A
SCHEMBL2135449 0.80 SLC10A2 (0.46) SLC10A2SLC10A1SLC10A6KMT2AGAA
SCHEMBL2138437 0.79 CCR1 (0.41) SLC10A2SLC10A1SLC10A6CYP3A4POLB
SCHEMBL16239807 0.79 FFAR4 (0.45) KMT2AGAAMEN1SLC22A12LMNA
SCHEMBL16239957 0.78 MCOLN2 (0.39) KMT2ATSHRLMNANPSR1SLC40A1
SCHEMBL16239801 0.78 MEN1 (0.50) KMT2AGAAMEN1TSHRPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2630124-B1 TETRAHYDROQUINOLINE DERIVATIVES USED AS AMPK ACTIVATORS HOFFMANN LA ROCHE (CH) 2014-11-19 EP claimed