SCHEMBL16239649

SCHEMBL16239649

CC1(C)CC(c2ccccc2NS(=O)(=O)c2ccccc2)Nc2c(C(F)(F)F)cccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.41
GAA P10253 2/20 0.41
SLC40A1 Q9NP59 3/20 0.39
FFAR4 Q5NUL3 1/20 0.37
RBP4 P02753 1/20 0.37
HTR6 P50406 2/20 0.35
MEN1 O00255 3/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
TSHR P16473 1/20 0.35
CYP2C19 P33261 1/20 0.35
MCOLN2 Q8IZK6 1/20 0.35
MCOLN3 Q8TDD5 1/20 0.35
MCOLN1 Q9GZU1 1/20 0.35
DDX3X O00571 2/20 0.35
ALDH1A1 P00352 2/20 0.34
RECQL P46063 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
SLC22A12 Q96S37 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16239499 0.93 KMT2A (0.41) KMT2AGAAFFAR4MEN1TSHR
SCHEMBL16239491 0.92 SLC10A2 (0.38) KMT2AGAASLC40A1MEN1CYP1A2
SCHEMBL16239817 0.88 SLC22A12 (0.47) KMT2ASLC40A1MEN1CYP1A2CYP3A4
SCHEMBL16239957 0.86 MCOLN2 (0.39) KMT2ASLC40A1TSHRMCOLN2MCOLN3
SCHEMBL16240077 0.85 TSHR (0.38) KMT2AGAASLC40A1HTR6MEN1
SCHEMBL16239807 0.83 FFAR4 (0.45) KMT2AGAAFFAR4HTR6MEN1
SCHEMBL16239675 0.82 HTR6 (0.35) SLC40A1HTR6MCOLN2MCOLN3MCOLN1
SCHEMBL16239801 0.80 MEN1 (0.50) KMT2AGAAMEN1TSHRMCOLN3
SCHEMBL2135223 0.80 LMNA (0.42) KMT2AGAASLC40A1MEN1ALDH1A1
SCHEMBL16239852 0.78 SLC10A2 (0.39) KMT2AGAAMEN1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2630124-B1 TETRAHYDROQUINOLINE DERIVATIVES USED AS AMPK ACTIVATORS HOFFMANN LA ROCHE (CH) 2014-11-19 EP claimed