SCHEMBL1624124

SCHEMBL1624124

O=C(O)NC(Cc1ccccc1)[C@@H]1CCNC1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 1/20 0.42
JAK3 P52333 1/20 0.41
CTSC P53634 1/20 0.41
LMNA P02545 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
MC4R P32245 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 2/20 0.39
SLC6A3 Q01959 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1624127 1.00 SMYD3 (0.42) SMYD3JAK3CTSCLMNATDP1
Hydrochloric Acid SCHEMBL1623813 0.91 CTSC (0.44) JAK3CTSCTDP1
Hydrochloric Acid SCHEMBL1623808 0.91 CTSC (0.44) JAK3CTSCTDP1
SCHEMBL6369980 0.85 PARP1 (0.40) SMYD3JAK3CTSCLMNATDP1
SCHEMBL3372476 0.85 LMNA (0.49) LMNATDP1NPC1RAB9AL3MBTL1
SCHEMBL5378282 0.83 CTSL (0.42) NPC1RAB9A
SCHEMBL3289149 0.82 ATM (0.50)
SCHEMBL5780237 0.82 ATM (0.50)
SCHEMBL27533342 0.82 ATM (0.50)
SCHEMBL4923835 0.81 TAAR1 (0.43) SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8283354-B2 Voltage gated sodium and calcium channel inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-10-09 US disclosed
US-7928107-B2 Quinazolines useful as modulators of ion channels VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-04-19 US disclosed
US-20060173018-A1 Quinazolines useful as modulators of ion channels VERTEX PHARMACEUTICALS INCORPORATED 2006-08-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060173018-A1 Quinazolines useful as modulators of ion channels KCNQ1, KCNQ2, KCNN3 SMYD3 1884/4885JAK3 3738/4885CTSC 1943/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.