SCHEMBL16277196

SCHEMBL16277196

Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)(C)C)cc1

nearest known ligand 0.80

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
VHL P40337 20/20 0.80
ELOC Q15369 11/20 0.80
ELOB Q15370 11/20 0.80

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17951935 1.00 VHL (0.80) VHLELOCELOB
SCHEMBL29843244 1.00 VHL (0.80) VHLELOCELOB
SCHEMBL19888885 1.00 VHL (0.80) VHLELOCELOB
SCHEMBL18090250 1.00 VHL (0.80) VHLELOCELOB
SCHEMBL19875334 1.00 VHL (0.80) VHLELOCELOB
SCHEMBL23098441 1.00 VHL (0.80) VHLELOCELOB
SCHEMBL18088944 0.94 VHL (0.73) VHLELOCELOB
SCHEMBL22291850 0.94 VHL (0.73) VHLELOCELOB
SCHEMBL22291849 0.93 VHL (0.77) VHLELOCELOB
SCHEMBL18063871 0.93 VHL (0.77) VHLELOCELOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 151 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4629981-A2 SMALL MOLECULE DEGRADERS OF C-SRC KINASE The Regents Of The University Of Michigan (US) 2025-10-15 EP claimed
WO-2024145315-A1 TARGETED PROTEIN DEGRADERS OF INDOLEAMINE 2,3-DIOXYGENASE 1 (IDO1) NORTHWESTERN UNIVERSITY (US) 2024-07-04 WO claimed
WO-2024123819-A2 SMALL MOLECULE DEGRADERS OF C-SRC KINASE THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2024-06-13 WO claimed
US-20220023431-A1 PROTEOLYSIS-TARGETING CHIMERIC MOLECULES (PROTACS) THAT INDUCE DEGRADATION OF INDOLEAMINE 2,3-DIOXYGENASE (IDO) PROTEIN NORTHWESTERN UNIVERSITY 2022-01-27 US claimed
US-20260131010-A1 MENIN PROTEOLYSIS TARGETING CHIMERAS (PROTACS) UNIV TEXAS (US) 2026-05-14 US disclosed
US-20260115296-A1 COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF RAPIDLY ACCELERATED FIBROSARCOMA POLYPEPTIDES UNIV YALE (US) 2026-04-30 US disclosed
EP-3886904-B1 IRAK DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS INC (US) 2026-04-22 EP disclosed
US-12569464-B2 Protein-protein interaction inducing technology ARVINAS OPERATIONS, INC. (US) 2026-03-10 US disclosed
US-12552783-B2 Modulators of proteolysis and associated methods of use ARVINAS OPERATIONS, INC. (US) 2026-02-17 US disclosed
US-12491252-B2 Substituted 3-amino-5-phenylbenzamide compounds as covalent inhibitors of enhancer zeste homolog 2 (EZH2) and proteolysis-targeting chimeric derivatives thereof (PROTACs) that induce degradation of EZH2 NORTHWESTERN UNIVERSITY (US) 2025-12-09 US disclosed
US-12492209-B2 Substituted [1,2,4]triazolo[4,3-c]pyrimidines that induce degradation of embryonic ectoderm development (EED) protein NORTHWESTERN UNIVERSITY (US) 2025-12-09 US disclosed
US-20250325673-A1 IRAK DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS INC (US) 2025-10-23 US disclosed
US-20170065719-A1 COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF BROMODOMAIN-CONTAINING PROTEINS ARVINAS OPERATIONS, INC. 2017-03-09 US disclosed
WO-2017030814-A1 COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF BROMODOMAIN-CONTAINING PROTEINS Arvinas, Inc. (US) 2017-02-23 WO disclosed
WO-2017030814-A1 COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF BROMODOMAIN-CONTAINING PROTEINS Arvinas, Inc. (US) 2017-02-23 WO disclosed
WO-2017011371-A1 MDM2-BASED MODULATORS OF PROTEOLYSIS AND ASSOCIATED METHODS OF USE ARVINAS, INC (US) 2017-01-19 WO disclosed
WO-2016146985-A1 DERIVATIVES OF 1-[(CYCLOPENTYL OR 2-PYRROLIDINYL)CARBONYLAMINOMETHYL]-4-(1,3-THIAZOL-5-YL) BENZENE WHICH ARE USEFUL FOR THE TREATMENT OF PROLIFERATIVE, AUTOIMMUNE OR INFLAMMATORY DISEASES UNIVERSITY OF DUNDEE (GB) 2016-09-22 WO disclosed
US-20160214972-A1 COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF ANDROGEN RECEPTOR ARVINAS OPERATIONS, INC. 2016-07-28 US disclosed
US-20160045607-A1 ESTROGEN-RELATED RECEPTOR ALPHA BASED PROTAC COMPOUNDS AND ASSOCIATED METHODS OF USE YALE UNIVERSITY 2016-02-18 US disclosed
US-20140356322-A1 Compounds & Methods for the Enhanced Degradation of Targeted Proteins & Other Polypeptides by an E3 Ubiquitin Ligase GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2014-12-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (12 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250325673-A1 IRAK DEGRADERS AND USES THEREOF IRAK2, IRAK3, IRAK1 VHL 2471/4885ELOC 874/4885ELOB 451/4885
US-20160214972-A1 COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF ANDROGEN RECEPTOR AR, ESRRA, MDM2 VHL 9/4885ELOC 411/4885ELOB 434/4885
US-20140356322-A1 Compounds & Methods for the Enhanced Degradation of Targeted Proteins & Other Polypeptides by an E3 Ubiquitin Ligase VHL, MDM2, STUB1 VHL 1/4885ELOC 190/4885ELOB 241/4885
US-20260131010-A1 MENIN PROTEOLYSIS TARGETING CHIMERAS (PROTACS) CRBN, UBE3C, PSME3 VHL 72/4885ELOC 136/4885ELOB 432/4885
US-12492209-B2 Substituted [1,2,4]triazolo[4,3-c]pyrimidines that induce degradation of embryonic ectoderm development (EED) protein EED, CUL3, PSME3 VHL 2296/4885ELOC 42/4885ELOB 274/4885
US-12569464-B2 Protein-protein interaction inducing technology STUB1, MDM2, XIAP VHL 1421/4885ELOC 1029/4885ELOB 980/4885
US-20220023431-A1 PROTEOLYSIS-TARGETING CHIMERIC MOLECULES (PROTACS) THAT INDUCE DEGRADATION OF INDOLEAMINE 2,3-DIOXYGENASE (IDO) PROTEIN IDO1, IDO2, KMO VHL 2395/4885ELOC 926/4885ELOB 2065/4885
US-12552783-B2 Modulators of proteolysis and associated methods of use CRBN, ADRM1, MDM2 VHL 37/4885ELOC 2051/4885ELOB 1657/4885
US-12491252-B2 Substituted 3-amino-5-phenylbenzamide compounds as covalent inhibitors of enhancer zeste homolog 2 (EZH2) and proteolysis-targeting chimeric derivatives thereof (PROTACs) that induce degradation of EZH2 EZH2, BAZ2A, BAZ2B VHL 235/4885ELOC 514/4885ELOB 183/4885
US-20160045607-A1 ESTROGEN-RELATED RECEPTOR ALPHA BASED PROTAC COMPOUNDS AND ASSOCIATED METHODS OF USE GPER1, PSMA3, ESR2 VHL 7/4885ELOC 153/4885ELOB 325/4885
US-20260115296-A1 COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF RAPIDLY ACCELERATED FIBROSARCOMA POLYPEPTIDES CRBN, VHL, ADRM1 VHL 2/4885ELOC 1043/4885ELOB 797/4885
US-20170065719-A1 COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF BROMODOMAIN-CONTAINING PROTEINS BRPF3, STUB1, BRDT VHL 11/4885ELOC 251/4885ELOB 223/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.