SCHEMBL16319655

SCHEMBL16319655

CS(=O)(=O)NC(=O)c1ccc(Oc2ccc(Cl)c(C(F)(F)F)c2)c(C#N)c1

nearest known ligand 0.62

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PLA2G7 Q13093 12/20 0.62
SCN9A Q15858 7/20 0.59
SCN5A Q14524 1/20 0.59
AR P10275 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16319487 0.88 SCN9A (0.65) PLA2G7SCN9ASCN5A
SCHEMBL16319332 0.88 SCN9A (0.61) PLA2G7SCN9ASCN5A
SCHEMBL16319499 0.86 SCN9A (0.63) PLA2G7SCN9ASCN5A
SCHEMBL16319828 0.85 SCN9A (0.70) SCN9ASCN5A
SCHEMBL371116 0.83 SCN9A (0.67) SCN9ASCN5A
SCHEMBL16319644 0.82 AR (0.58) PLA2G7SCN9ASCN5AAR
SCHEMBL679345 0.82 SCN9A (0.51) PLA2G7SCN9ASCN5A
SCHEMBL680479 0.82 SCN9A (0.50) PLA2G7SCN9ASCN5AAR
SCHEMBL16319531 0.81 SCN9A (0.58) SCN9ASCN5A
SCHEMBL679917 0.80 SCN9A (0.50) PLA2G7SCN9ASCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593427-B1 SULFONAMIDE DERIVATIVES AS NAV1.7 INHIBITORS FOR THE TREATMENT OF PAIN PFIZER LTD (GB) 2014-12-24 EP disclosed