SCHEMBL16333641

SCHEMBL16333641

Cc1onc(-c2cccnc2)c1C(=O)O

nearest known ligand 0.63

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.63
POLB P06746 2/20 0.63
KDM4E B2RXH2 1/20 0.63
L3MBTL1 Q9Y468 1/20 0.63
GAA P10253 2/20 0.56
KMT2A Q03164 2/20 0.56
MEN1 O00255 1/20 0.56
LMNA P02545 1/20 0.55
SMN1; SMN2 Q16637 2/20 0.53
MAPK1 P28482 1/20 0.53
TSHR P16473 3/20 0.48
HTT P42858 2/20 0.48
GABRA5 P31644 1/20 0.47
USP2 O75604 1/20 0.47
MKNK1 Q9BUB5 1/20 0.46
MKNK2 Q9HBH9 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12542895 0.91 ALDH1A1 (0.57) ALDH1A1POLBKDM4EL3MBTL1GAA
SCHEMBL12544175 0.89 ALDH1A1 (0.58) ALDH1A1POLBKDM4EL3MBTL1GAA
SCHEMBL316093 0.84 KMT2A (0.76) ALDH1A1POLBGAAKMT2AMEN1
Hydrochloric Acid SCHEMBL4846563 0.83 KMT2A (0.73) ALDH1A1POLBGAAKMT2AMEN1
SCHEMBL12543204 0.83 KMT2A (0.51) ALDH1A1POLBKDM4EL3MBTL1GAA
SCHEMBL2930011 0.82 POLB (0.63) ALDH1A1POLBKDM4EL3MBTL1GAA
SCHEMBL6315186 0.82 TDO2 (0.49) ALDH1A1POLBKDM4EL3MBTL1GAA
SCHEMBL6069148 0.81 SMN1; SMN2 (0.62) ALDH1A1POLBKDM4EL3MBTL1GAA
SCHEMBL5424589 0.80 MKNK1 (0.58) ALDH1A1POLBKDM4EL3MBTL1GAA
SCHEMBL23830221 0.79 ALDH1A1 (0.47) ALDH1A1POLBKDM4EL3MBTL1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2227467-B1 ISOXAZOLO-PYRIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2014-12-31 EP disclosed
CN-101346372-B Aryl-isoxazol-4-yl-oxadiazole derivatives HOFFMANN LA ROCHE 2011-09-28 CN disclosed
CN-101346372-A Aryl-isoxazol-4-yl-oxadiazole derivatives HOFFMANN LA ROCHE (CH) 2009-01-14 CN disclosed