SCHEMBL163387

SCHEMBL163387

Cc1ccc2[c]nc(C(=O)c3ccc(F)cc3)nc2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.39
GAA P10253 1/20 0.39
GRM2 Q14416 1/20 0.38
HSD17B14 Q9BPX1 1/20 0.38
KMT2A Q03164 3/20 0.38
HTT P42858 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 3/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
ALDH1A1 P00352 2/20 0.37
TDP1 Q9NUW8 1/20 0.37
KCNMA1 Q12791 1/20 0.37
F2 P00734 1/20 0.37
PLAU P00749 1/20 0.37
ELANE P08246 1/20 0.37
PAX8 Q06710 1/20 0.36
LTA4H P09960 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
PTGS1 P23219 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL164593 0.75 GRM2 (0.47) GRM5GAAGRM2HSD17B14KMT2A
SCHEMBL2966992 0.67 ALDH1A1 (0.76) KMT2AHTTMEN1LMNASMN1; SMN2
SCHEMBL14407932 0.67 ALDH1A1 (0.76) KMT2AHTTMEN1LMNASMN1; SMN2
SCHEMBL15888794 0.66 ALDH1A1 (0.59) KMT2AHTTMEN1LMNASMN1; SMN2
SCHEMBL7811187 0.66 SMN1; SMN2 (0.68) HTTLMNASMN1; SMN2ALDH1A1TDP1
SCHEMBL1584825 0.66 F2 (0.59) GAAKMT2AHTTLMNASMN1; SMN2
SCHEMBL6097936 0.64 MAPT (0.49) KMT2AHTTMEN1LMNASMN1; SMN2
SCHEMBL14099187 0.64 LMNA (0.50) KMT2AHTTLMNASMN1; SMN2ALDH1A1
SCHEMBL17716230 0.64 KMT2A (0.64) GAAKMT2AHTTKDM4EMEN1
SCHEMBL15679982 0.64 CES2 (0.76) GAAKMT2AHTTMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611502-A1 ADENOSINE A3 RECEPTOR MODULATING COMPOUNDS AND METHODS OF USE THEREOF Ambit Biosciences Corporation (US) 2013-07-10 EP disclosed
WO-2012030918-A1 ADENOSINE A3 RECEPTOR MODULATING COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2012-03-08 WO disclosed