SCHEMBL16338973

SCHEMBL16338973

Cc1ccc2o[c]cc2n1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.39
CCR1 P32246 1/20 0.34
RAB9A P51151 1/20 0.34
CCR5 P51681 1/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
POLB P06746 1/20 0.34
CASP6 P55212 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7512293 0.66 CYP1A2 (0.59) CYP1A2CCR1RAB9ACCR5KDM4E
SCHEMBL8312831 0.65 DYRK1A (0.46) CYP1A2CCR1RAB9ACCR5KDM4E
SCHEMBL207520 0.64 CYP2A6 (0.44) CYP1A2RAB9AKDM4E
SCHEMBL7916567 0.64 CYP1A2 (0.48) CYP1A2RAB9AKDM4ELMNAPOLB
SCHEMBL8337485 0.64 CYP1A2 (0.40) CYP1A2CCR1RAB9ACCR5KDM4E
SCHEMBL9217980 0.62 CYP1A2 (0.65) CYP1A2CCR1RAB9ACCR5KDM4E
SCHEMBL25244668 0.62 CCR1 (0.34) CYP1A2CCR1RAB9ACCR5
SCHEMBL1165531 0.61 CYP1A2 (0.41) CYP1A2RAB9AKDM4ELMNAPOLB
SCHEMBL30528375 0.61 CYP1A2 (0.41) CYP1A2RAB9AKDM4ELMNAPOLB
SCHEMBL295035 0.61 CYP1A2 (0.54) CYP1A2CCR1RAB9ACCR5KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 48 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111182898-B Methods for treating huntington's disease PTC医疗公司 2024-04-16 CN disclosed
US-20240067646-A1 COMPOUNDS FOR TREATING SPINAL MUSCULAR ATROPHY HOFFMANN-LA ROCHE INC. 2024-02-29 US disclosed
US-20230310651-A1 METHODS FOR MODULATING RNA SPLICING PTC THERAPEUTICS, INC. (US) 2023-10-05 US disclosed
EP-4249472-A2 METHODS FOR MODULATING RNA SPLICING PTC Therapeutics, Inc. (US) 2023-09-27 EP disclosed
US-11753407-B2 Compounds for treating spinal muscular atrophy PTC THERAPEUTICS, INC. (US) 2023-09-12 US disclosed
US-20230272367-A1 METHODS FOR MODULATING RNA SPLICING PTC THERAPEUTICS, INC. (US) 2023-08-31 US disclosed
EP-3644996-B1 METHODS FOR TREATING HUNTINGTON'S DISEASE PTC THERAPEUTICS INC (US) 2023-07-26 EP disclosed
US-11702646-B2 Methods for modulating RNA splicing PTC THERAPEUTICS, INC. (US) 2023-07-18 US disclosed
EP-3310169-B1 METHODS FOR MODULATING RNA SPLICING PTC THERAPEUTICS INC (US) 2023-05-17 EP disclosed
US-11602567-B2 Methods for modulating RNA splicing PTC THERAPEUTICS, INC. (US) 2023-03-14 US disclosed
US-9617268-B2 Compounds for treating spinal muscular atrophy PTC THERAPEUTICS, INC. (US) 2017-04-11 US disclosed
US-9586955-B2 Compounds for treating spinal muscular atrophy PTC THERAPEUTICS, INC. (US) 2017-03-07 US disclosed
US-20170000794-A1 METHODS FOR MODULATING THE AMOUNT OF RNA TRANSCRIPTS PTC THERAPEUTICS, INC. 2017-01-05 US disclosed
US-9399649-B2 Compounds for treating spinal muscular atrophy PTC THERAPEUTICS, INC. (US) 2016-07-26 US disclosed
US-9371336-B2 Compounds for treating spinal muscular atrophy PTC THERAPEUTICS, INC. (US) 2016-06-21 US disclosed
US-20150166575-A1 COMPOUNDS FOR TREATING SPINAL MUSCULAR ATROPHY PTC THERAPEUTICS INC. (US) 2015-06-18 US disclosed
US-20150126515-A1 COMPOUNDS FOR TREATING SPINAL MUSCULAR ATROPHY PTC THERAPEUTICS, INC. (US) 2015-05-07 US disclosed
US-20150119380-A1 COMPOUNDS FOR TREATING SPINAL MUSCULAR ATROPHY F. HOFFMANN-LA ROCHE AG (CH) 2015-04-30 US disclosed
US-20150080383-A1 COMPOUNDS FOR TREATING SPINAL MUSCULAR ATROPHY PTC THERAPEUTICS, INC. 2015-03-19 US disclosed
US-20150005289-A1 COMPOUNDS FOR TREATING SPINAL MUSCULAR ATROPHY HOFFMANN-LA ROCHE INC. 2015-01-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (12 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240067646-A1 COMPOUNDS FOR TREATING SPINAL MUSCULAR ATROPHY SMN1; SMN2, CPT1B, GYS1 CYP1A2 4324/4885CCR1 4016/4885RAB9A 1350/4885
US-20150005289-A1 COMPOUNDS FOR TREATING SPINAL MUSCULAR ATROPHY SMN1; SMN2, CPT1B, GYS1 CYP1A2 4663/4885CCR1 4266/4885RAB9A 1728/4885
US-20230272367-A1 METHODS FOR MODULATING RNA SPLICING RBM17, SNRPE, HNRNPM CYP1A2 4151/4885CCR1 4765/4885RAB9A 2369/4885
US-20150080383-A1 COMPOUNDS FOR TREATING SPINAL MUSCULAR ATROPHY SMN1; SMN2, CPT1B, GYS1 CYP1A2 4663/4885CCR1 4266/4885RAB9A 1728/4885
US-20150126515-A1 COMPOUNDS FOR TREATING SPINAL MUSCULAR ATROPHY SMN1; SMN2, CPT1B, GYS1 CYP1A2 4663/4885CCR1 4266/4885RAB9A 1728/4885
US-11702646-B2 Methods for modulating RNA splicing RBM17, SNRPE, HNRNPM CYP1A2 4151/4885CCR1 4765/4885RAB9A 2369/4885
US-20150119380-A1 COMPOUNDS FOR TREATING SPINAL MUSCULAR ATROPHY SMN1; SMN2, RBM17, RBM22 CYP1A2 4539/4885CCR1 3824/4885RAB9A 3292/4885
US-11602567-B2 Methods for modulating RNA splicing RBM17, SNRPE, RBM3 CYP1A2 4330/4885CCR1 4741/4885RAB9A 2689/4885
US-20170000794-A1 METHODS FOR MODULATING THE AMOUNT OF RNA TRANSCRIPTS RNMT, NSUN2, RNGTT CYP1A2 4410/4885CCR1 4277/4885RAB9A 3864/4885
US-20150166575-A1 COMPOUNDS FOR TREATING SPINAL MUSCULAR ATROPHY SMN1; SMN2, CPT1B, GYS1 CYP1A2 4663/4885CCR1 4266/4885RAB9A 1728/4885
US-20230310651-A1 METHODS FOR MODULATING RNA SPLICING RBM17, SNRPE, RBM3 CYP1A2 4330/4885CCR1 4741/4885RAB9A 2689/4885
US-11753407-B2 Compounds for treating spinal muscular atrophy SMN1; SMN2, CPT1B, GYS1 CYP1A2 4094/4885CCR1 3356/4885RAB9A 1386/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.