SCHEMBL16396113

SCHEMBL16396113

CS(=O)(=O)Nc1c(C(N)=O)sc2ccccc12

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LIMK1 P53667 2/20 0.68
ACLY P53396 1/20 0.60
IKBKB O14920 1/20 0.54
KDM4E B2RXH2 3/20 0.46
ALDH1A1 P00352 2/20 0.46
HSD17B10 Q99714 2/20 0.46
MEN1 O00255 1/20 0.46
GLA P06280 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
HPGD P15428 1/20 0.46
ALOX15 P16050 1/20 0.46
KMT2A Q03164 1/20 0.46
ATM Q13315 1/20 0.46
LMNA P02545 1/20 0.43
MAPK1 P28482 1/20 0.43
OGG1 O15527 1/20 0.42
HSD11B1 P28845 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC8 Q9BY41 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13969608 0.81 LIMK1 (1.00) LIMK1ACLYIKBKBKDM4EALDH1A1
SCHEMBL5809803 0.80 ACLY (0.45) LIMK1ACLYLMNAMAPK1HSD11B1
SCHEMBL18088617 0.76 KEAP1 (0.42) LIMK1ACLYALDH1A1EP300KAT2B
SCHEMBL2702750 0.73 LIMK1 (0.68) LIMK1ACLYIKBKBKDM4EALDH1A1
SCHEMBL29483598 0.73 LIMK1 (0.68) LIMK1ACLYIKBKBKDM4EALDH1A1
SCHEMBL9433865 0.72 LIMK1 (0.62) LIMK1ACLYIKBKBKDM4EALDH1A1
SCHEMBL6609258 0.71 LIMK1 (1.00) LIMK1IKBKBKDM4EALDH1A1HSD17B10
SCHEMBL11074064 0.71 LIMK1 (0.68) LIMK1ACLYIKBKBKDM4EALDH1A1
SCHEMBL649968 0.71 LIMK1 (0.68) LIMK1ACLYIKBKBKDM4EALDH1A1
SCHEMBL29604679 0.70 LIMK1 (0.58) LIMK1ACLYIKBKBHSD17B10LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3004057-A1 HETEROCYCLIC DERIVATIVES AND USE THEREOF C&C Research Laboratories (KR) 2016-04-13 EP claimed
WO-2014196793-A1 HETEROCYCLIC DERIVATIVES AND USE THEREOF C&C RESEARCH LABORATORIES (KR) 2014-12-11 WO claimed
EP-3004057-A1 HETEROCYCLIC DERIVATIVES AND USE THEREOF C&C Research Laboratories (KR) 2016-04-13 EP disclosed
WO-2014196793-A1 HETEROCYCLIC DERIVATIVES AND USE THEREOF C&C RESEARCH LABORATORIES (KR) 2014-12-11 WO disclosed