SCHEMBL16396184

SCHEMBL16396184

COc1ccc(COC(=O)c2cc(OCc3ccc(OC)cc3)cc([N+](=O)[O-])c2)cc1.O=C(O)c1cc(O)cc([N+](=O)[O-])c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.51
RAB9A P51151 3/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
NPC1 O15118 1/20 0.49
POLB P06746 1/20 0.49
PLA2G4B P0C869 2/20 0.47
MAPT P10636 2/20 0.46
ALDH1A1 P00352 2/20 0.46
GAA P10253 1/20 0.45
MAOB P27338 3/20 0.45
MAOA P21397 1/20 0.44
TP53 P04637 1/20 0.43
PKM P14618 1/20 0.43
NFKB1 P19838 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
MRGPRX4 Q96LA9 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16396138 0.92 HTT (0.59) HTTRAB9ASMN1; SMN2NPC1POLB
SCHEMBL16396254 0.89 RAB9A (0.60) RAB9ASMN1; SMN2NPC1POLBPLA2G4B
SCHEMBL417705 0.81 MAPT (0.60) HTTRAB9AMAPTALDH1A1MAOB
SCHEMBL16396350 0.80 MAOB (0.53) RAB9ASMN1; SMN2NPC1POLBPLA2G4B
SCHEMBL11265699 0.78 MEN1 (0.70) RAB9APLA2G4BMAPTALDH1A1MAOB
SCHEMBL8403461 0.76 ALDH1A1 (0.65) HTTRAB9ASMN1; SMN2NPC1POLB
SCHEMBL8561986 0.75 KMT2A (0.55) HTTRAB9ANPC1MAPTALDH1A1
SCHEMBL1107602 0.74 SMPD1 (0.56) HTTRAB9ASMN1; SMN2NPC1POLB
SCHEMBL1099548 0.73 MEN1 (0.55) HTTRAB9ASMN1; SMN2NPC1MAPT
SCHEMBL6841271 0.72 MAPT (0.53) POLBMAPTALDH1A1MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3004057-A1 HETEROCYCLIC DERIVATIVES AND USE THEREOF C&C Research Laboratories (KR) 2016-04-13 EP disclosed
WO-2014196793-A1 HETEROCYCLIC DERIVATIVES AND USE THEREOF C&C RESEARCH LABORATORIES (KR) 2014-12-11 WO disclosed