SCHEMBL16455992

SCHEMBL16455992

CC(C)(C)c1ccc(-n2c(=O)oc3ccccc32)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNKS O95271 1/20 0.50
MAPK1 P28482 3/20 0.44
TSHR P16473 2/20 0.44
HPGD P15428 2/20 0.44
USP2 O75604 1/20 0.44
ALDH1A1 P00352 5/20 0.41
NPSR1 Q6W5P4 3/20 0.41
MIF P14174 1/20 0.40
GAA P10253 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PMM2 O15305 1/20 0.39
MPI P34949 1/20 0.39
PHOSPHO1 Q8TCT1 1/20 0.39
IDO1 P14902 2/20 0.39
LMNA P02545 1/20 0.39
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
PIK3CD O00329 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CB P42338 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15289179 0.82 ALDH1A1 (0.56) TNKSMAPK1TSHRHPGDUSP2
SCHEMBL4622801 0.81 TNKS (0.55) TNKSMAPK1TSHRHPGDUSP2
SCHEMBL24703353 0.79 KDM4E (0.44) TNKSMAPK1HPGDALDH1A1NPSR1
SCHEMBL16456377 0.78 MAPK1 (0.50) TNKSMAPK1TSHRHPGDUSP2
SCHEMBL14580062 0.74 TNKS (0.49) TNKSMAPK1TSHRHPGDUSP2
SCHEMBL24703436 0.73 KDM4E (0.57) MAPK1TSHRALDH1A1NPSR1PMM2
SCHEMBL674884 0.71 KDM4E (0.59) MAPK1TSHRALDH1A1NPSR1PMM2
SCHEMBL29875801 0.71 KDM4E (0.59) MAPK1TSHRALDH1A1NPSR1PMM2
SCHEMBL12049010 0.71 MAPK1 (0.53) MAPK1TSHRHPGDUSP2ALDH1A1
SCHEMBL4004493 0.70 TNKS (0.43) TNKSMAPK1TSHRHPGDUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9340549-B2 Oxazolidinone compounds and derivatives thereof AMGEN INC. (US) 2016-05-17 US disclosed
US-20150045368-A1 OXAZOLIDINONE COMPOUNDS AND DERIVATIVES THEREOF AMGEN INC. 2015-02-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150045368-A1 OXAZOLIDINONE COMPOUNDS AND DERIVATIVES THEREOF TNKS1BP1, TNKS, TBKBP1 TNKS 2/4885MAPK1 1337/4885TSHR 3044/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.