SCHEMBL16474145

SCHEMBL16474145

Nn1[nH]c2ccccc2c1=O

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.59
MPI P34949 1/20 0.57
ALDH1A1 P00352 2/20 0.55
TRPV1 Q8NER1 1/20 0.46
ADORA3 P0DMS8 1/20 0.46
ADORA2A P29274 1/20 0.46
ADORA2B P29275 1/20 0.46
ADORA1 P30542 1/20 0.46
CA12 O43570 1/20 0.46
RNASEH1 O60930 1/20 0.46
ERCC1 P07992 1/20 0.46
ERCC5 P28715 1/20 0.46
FEN1 P39748 1/20 0.46
CA9 Q16790 1/20 0.46
ERCC4 Q92889 1/20 0.46
KDM4E B2RXH2 1/20 0.44
GLA P06280 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL189858 0.78 KDM4E (0.59) ALOX5MPIALDH1A1KDM4E
SCHEMBL29930611 0.78 KDM4E (0.59) ALOX5MPIALDH1A1KDM4E
SCHEMBL1316369 0.77 KDM4E (0.57) ALOX5MPIALDH1A1CA12CA9
SCHEMBL1316368 0.77 KDM4E (0.57) ALOX5MPIALDH1A1KDM4E
SCHEMBL30336436 0.74 ALOX5 (1.00) ALOX5MPIADORA3ADORA2AADORA2B
SCHEMBL2673327 0.74 ALOX5 (1.00) ALOX5MPIADORA3ADORA2AADORA2B
SCHEMBL17750809 0.74 ALOX5 (0.59) ALOX5MPIALDH1A1TRPV1ADORA3
SCHEMBL2438599 0.72 MPI (1.00) ALOX5MPITRPV1
SCHEMBL30423726 0.72 MPI (1.00) ALOX5MPITRPV1
SCHEMBL5929408 0.72 ALOX5 (0.52) ALOX5MPIALDH1A1TRPV1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021224680-A1 SUBSTITUTED BENZOTRIAZINONE METABOLITES OF A GPR139 AGONIST TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2021-11-11 WO disclosed
EP-2406215-B1 OXO-HETEROCYCLICALLY SUBSTITUTED ALKYL CARBOXYLIC ACIDS AND USE THEREOF BAYER IP GMBH (DE) 2014-04-16 EP disclosed