SCHEMBL1316368

SCHEMBL1316368

Nn1[nH]c(=O)c2ccccc2c1=O.[NaH]

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.57
TP53 P04637 1/20 0.57
TSHR P16473 1/20 0.55
GAA P10253 2/20 0.47
MAPK1 P28482 2/20 0.47
GLS O94925 1/20 0.47
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
POLB P06746 1/20 0.44
PLEC Q15149 1/20 0.44
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
ALDH1A1 P00352 3/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 1/20 0.41
HPGD P15428 1/20 0.41
CYP2C19 P33261 1/20 0.41
ALOX5 P09917 1/20 0.38
TNKS O95271 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29930611 0.98 KDM4E (0.59) KDM4ETP53TSHRGAAMAPK1
SCHEMBL189858 0.98 KDM4E (0.59) KDM4ETP53TSHRGAAMAPK1
SCHEMBL1316369 0.96 KDM4E (0.57) KDM4ETP53TSHRGAAMAPK1
SCHEMBL16474145 0.77 ALOX5 (0.59) KDM4EALDH1A1ALOX5MPI
SCHEMBL194708 0.77 KDM4E (0.44) KDM4ETP53TSHRGAAMAPK1
SCHEMBL19577293 0.74 KDM4E (0.61) KDM4ETP53TSHRGAAMAPK1
SCHEMBL7070837 0.73 KDM4E (0.42) KDM4ETP53TSHRGAAMEN1
SCHEMBL1618278 0.72 KDM4E (0.59) KDM4ETP53TSHRGAAMAPK1
SCHEMBL31091767 0.72 KDM4E (1.00) KDM4ETP53TSHRGAAMAPK1
SCHEMBL1101962 0.72 KDM4E (1.00) KDM4ETP53TSHRGAAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180153889-A1 MODULATION OF CELL FATES AND ACTIVITIES BY PHTHALAZINEDIONES BACH PHARMA, INC. 2018-06-07 US disclosed
US-9968602-B2 Modulation of cell fates and activities by phthalazinediones BACH PHARMA, INC. (US) 2018-05-15 US disclosed
CN-107567437-A Crystalline form of 5-amino-2, 3-dihydrophthalazine-1, 4-dione sodium salt, pharmaceutical preparation containing it and process for its production 麦翠奥制药公司 2018-01-09 CN disclosed
EP-2389364-B1 NEW METHOD FOR OBTAINING 5-AMINO-2,3-DIHYDROPHTHALAZINE-1,4-DIONE ALKALI METAL SALTS AND THEIR USE IN MEDICINE ABIDOPHARMA PL SP Z O O (PL) 2016-10-26 EP disclosed
US-9101629-B2 Method for obtaining 5-amino-2,3-dihydrophthalazine-1,4-dione alkali metal salts and their use in medicine ABIDOPHARMA PL SP. Z O.O. (PL) 2015-08-11 US disclosed
US-20140113902-A1 METHOD FOR OBTAINING 5-AMINO-2,3-DIHYDROPHTHALAZINE-1,4-DIONE ALKALI METAL SALTS AND THEIR USE IN MEDICINE Abidopharma PL SP. Z.O.O. (PL) 2014-04-24 US disclosed
US-20140030317-A1 MODULATION OF CELL FATES AND ACTIVITIES BY PHTHALAZINEDIONES Occhiuti & Rohlicek LLP 2014-01-30 US disclosed
US-8536171-B2 Method for obtaining 5-amino 2,3-dihydrophthalazine-1,4-dione alkali metal salts and their use in medicine Abidopharma PL SP. Z.O.O. (PL) 2013-09-17 US disclosed
EP-2389364-A2 NEW METHOD FOR OBTAINING 5-AMINO-2,3-DIHYDROPHTHALAZINE-1,4-DIONE ALKALI METAL SALTS AND THEIR USE IN MEDICINE Abidopharma Pl SP. Z.O.O (PL) 2011-11-30 EP disclosed
US-20110275642-A1 NEW METHOD FOR OBTAINING 5-AMINO 2,3-DIHYDROPHTHALAZINE-1,4-DIONE ALKALI METAL SALTS AND THEIR USE IN MEDICINE Abidopharma PL SP. Z.O.O. (PL) 2011-11-10 US disclosed
US-20090018137-A1 MODULATION OF CELL FATES AND ACTIVITIES BY PHTHALAZINEDIONES BACH PHARMA, INC. (US) 2009-01-15 US disclosed
EP-1924274-A4 MODULATION OF CELL FATES AND ACTIVITIES BY PHTHALAZINEDIONES BACH PHARMA INC (US) 2008-10-08 EP disclosed
EP-1924274-A1 MODULATION OF CELL FATES AND ACTIVITIES BY PHTHALAZINEDIONES Bach Pharma, Inc (US) 2008-05-28 EP disclosed
US-7326690-B2 Modulation of cell fates and activities by phthalazinediones BACH PHARMA, INC. (US) 2008-02-05 US disclosed
US-20070142303-A1 Modulation of cell fates and activities by phthalazinediones BACH PHARMA, INC. (US) 2007-06-21 US disclosed
WO-2007018546-A1 MODULATION OF CELL FATES AND ACTIVITIES BY PHTHALAZINEDIONES BACH PHARMA, INC. (US) 2007-02-15 WO disclosed
US-20050288291-A1 Modulation of cell fates and activities by phthalazinediones BACH PHARMA, INC. (US) 2005-12-29 US disclosed
US-20020198208-A1 MEDICINAL PREPARATION AND PROCESS FOR MANUFACTURING THEREOF ABIDOV, MUSA TAZHUDINOVICH (RU) 2002-12-26 US disclosed
US-6489326-B1 SODIUM NUCLEINATE, 2-AMINO-1,2,3,4-TETRAHYDROPHTHALAZINE-1,4-DIONE SODIUM SALT DIHYDRATE, USED AS AN IMMUNOMODULATOR, WHICH ALSO HAS ANTIINFLAMMATORY AND ANTIOXIDANT PROPERTIES Pavlov, Anatoliy Ivanovich (RU) 2002-12-03 US disclosed
EP-1203587-A1 A MEDICAMENT AND METHOD FOR THE PRODUCTION THEREOF Abidov, Musea Tazhudinovich (RU) 2002-05-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110275642-A1 NEW METHOD FOR OBTAINING 5-AMINO 2,3-DIHYDROPHTHALAZINE-1,4-DIONE ALKALI METAL SALTS AND THEIR USE IN MEDICINE ADH1C, SCN5A, ADH1A KDM4E 2263/4885TP53 2286/4885TSHR 3071/4885
US-20180153889-A1 MODULATION OF CELL FATES AND ACTIVITIES BY PHTHALAZINEDIONES NFE2L2, GPX4, TXNRD2 KDM4E 2063/4885TP53 89/4885TSHR 3785/4885
US-20140113902-A1 METHOD FOR OBTAINING 5-AMINO-2,3-DIHYDROPHTHALAZINE-1,4-DIONE ALKALI METAL SALTS AND THEIR USE IN MEDICINE SCN5A, SLC5A2, KCNJ2 KDM4E 1852/4885TP53 3567/4885TSHR 3013/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.