SCHEMBL1647896

SCHEMBL1647896

COc1cccc(CNC(=O)c2n[nH]c3cc(-c4ncnc5[nH]ccc45)ccc23)c1

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PRKACA P17612 3/20 0.65
PRKACG P22612 3/20 0.65
PRKACB P22694 3/20 0.65
SMN1; SMN2 Q16637 1/20 0.64
ROCK2 O75116 8/20 0.57
ROCK1 Q13464 3/20 0.49
MAPT P10636 2/20 0.49
BTK Q06187 2/20 0.49
TNIK Q9UKE5 1/20 0.47
PDGFRB P09619 1/20 0.47
KIT P10721 1/20 0.47
FLT3 P36888 1/20 0.47
MAP3K19 Q56UN5 1/20 0.47
JAK2 O60674 1/20 0.46
JAK1 P23458 1/20 0.46
TYK2 P29597 1/20 0.46
JAK3 P52333 1/20 0.46
RPS6KB1 P23443 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1647246 0.87 PRKACA (0.65) PRKACAPRKACGPRKACBSMN1; SMN2ROCK2
SCHEMBL12779514 0.84 BTK (0.52) PRKACAPRKACGPRKACBSMN1; SMN2BTK
SCHEMBL12779737 0.83 ROCK2 (0.67) PRKACAPRKACGPRKACBROCK2ROCK1
SCHEMBL1647171 0.83 PRKACA (0.61) PRKACAPRKACGPRKACBSMN1; SMN2ROCK2
SCHEMBL12779421 0.81 PRKACA (0.77) PRKACAPRKACGPRKACBSMN1; SMN2ROCK2
SCHEMBL13362826 0.79 MMP13 (0.51) ROCK2ROCK1MAPTBTKTNIK
SCHEMBL13457054 0.79 ROCK2 (0.64) ROCK2ROCK1BTKTNIKPDGFRB
SCHEMBL3128936 0.79 ROCK2 (0.62) ROCK2BTKPDGFRBKITFLT3
SCHEMBL1647780 0.79 PRKACA (1.00) PRKACAPRKACGPRKACBSMN1; SMN2ROCK2
SCHEMBL1648102 0.77 CLK1 (0.52) PRKACAPRKACGPRKACBSMN1; SMN2ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011050245-A1 BICYCLIC HETEROARYLS AS KINASE INHIBITORS FENG YANGBO (US) 2011-04-28 WO disclosed
WO-2011050245-A1 BICYCLIC HETEROARYLS AS KINASE INHIBITORS FENG YANGBO (US) 2011-04-28 WO disclosed