Hydrazine

Hydrazine

SCHEMBL1648713

COc1ccc(CC(C)C(=O)O)cc1OC.NN

nearest known ligand 0.71

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.71
ALOX15 P16050 3/20 0.54
ALOX12 P18054 2/20 0.54
PPARD Q03181 2/20 0.52
PPARA Q07869 2/20 0.52
MAPK1 P28482 1/20 0.51
MMP1 P03956 1/20 0.50
ALDH1A1 P00352 1/20 0.50
ATM Q13315 2/20 0.49
TUBB1 Q9H4B7 1/20 0.49
NPC1 O15118 1/20 0.49
LMNA P02545 1/20 0.49
HTT P42858 1/20 0.49
CA2 P00918 1/20 0.49
FOS P01100 1/20 0.47
TTR P02766 1/20 0.47
JUN P05412 1/20 0.47
NR3C1 P04150 1/20 0.47
HSD17B1 P14061 1/20 0.47
HSD17B2 P37059 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9781691 0.97 LDHA (0.76) LDHAALOX15ALOX12PPARDPPARA
SCHEMBL18082680 0.97 LDHA (0.76) LDHAALOX15ALOX12PPARDPPARA
SCHEMBL3175155 0.84 FOS (0.69) LDHAALOX15ALOX12MAPK1MMP1
SCHEMBL22108693 0.84 FOS (0.69) LDHAALOX15ALOX12MAPK1MMP1
SCHEMBL16913261 0.84 LDHA (0.58) LDHAALOX15ALOX12PPARDPPARA
SCHEMBL16973674 0.84 LDHA (0.66) LDHAALOX15ALOX12MAPK1ALDH1A1
SCHEMBL10734796 0.84 LDHA (0.66) LDHAALOX15ALOX12PPARDPPARA
SCHEMBL490731 0.83 LDHA (1.00) LDHAALOX15ALOX12MAPK1MMP1
SCHEMBL9518156 0.83 MMP1 (0.58) LDHAMMP1ALDH1A1NPC1HTT
SCHEMBL15570321 0.83 LDHA (0.56) LDHAPPARDPPARAMMP1TUBB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8491929-B2 Bioadhesive polymers VAUNNEX INC. (US) 2013-07-23 US disclosed
US-20110086095-A1 Bioadhesive Polymers Spherics, Inc (MA) 2011-04-14 US disclosed
US-20100316712-A1 PHARMACEUTICAL COMPOSITIONS FOR TREATMENT OF PARKINSON'S DISEASE AND RELATED DISORDERS COMBINATORX, INCORPORATED (US) 2010-12-16 US disclosed
US-20080299204-A1 Dosage forms for movement disorder treatment SPHERICS, INC. (US) 2008-12-04 US disclosed
US-20080131492-A1 Dosage forms for movement disorder treatment SPHERICS, INC. (US) 2008-06-05 US disclosed
EP-1901720-A2 IMPROVED DOSAGE FORMS FOR MOVEMENT DISORDER TREATMENT Spherics, Inc. (US) 2008-03-26 EP disclosed
WO-2008002471-A2 EROSION-STABILIZED BIOADHESIVE POLYMERS FUNCTIONALIZED OR BLENDED WITH CATECHOL AND DERIVATIVES THEREOF SPHERICS, INC. (US) 2008-01-03 WO disclosed
US-20070148238-A1 Dosage forms for movement disorder treatment SPHERICS, INC. (US) 2007-06-28 US disclosed
WO-2007002516-A2 IMPROVED DOSAGE FORMS FOR MOVEMENT DISORDER TREATMENT SPHERICS, INC. (US) 2007-01-04 WO disclosed
WO-2007002318-A2 BIOADHESIVE POLYMERS SPHERICS, INC. (US) 2007-01-04 WO disclosed
US-20070003621-A1 Dosage forms for movement disorder treatment SPHERICS, INC. (US) 2007-01-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110086095-A1 Bioadhesive Polymers CD44, EPCAM, ABCG2 LDHA 109/4885ALOX15 1971/4885ALOX12 1451/4885
US-20100316712-A1 PHARMACEUTICAL COMPOSITIONS FOR TREATMENT OF PARKINSON'S DISEASE AND RELATED DISORDERS PARK7, SNCA, COMT LDHA 560/4885ALOX15 317/4885ALOX12 544/4885
US-20070148238-A1 Dosage forms for movement disorder treatment PARK7, SNCA, HTT LDHA 1644/4885ALOX15 1133/4885ALOX12 1699/4885
US-20080131492-A1 Dosage forms for movement disorder treatment PARK7, SNCA, HTT LDHA 1644/4885ALOX15 1133/4885ALOX12 1699/4885
US-20070003621-A1 Dosage forms for movement disorder treatment PARK7, SNCA, HTT LDHA 1644/4885ALOX15 1133/4885ALOX12 1699/4885
US-20080299204-A1 Dosage forms for movement disorder treatment PARK7, SNCA, HTT LDHA 1644/4885ALOX15 1133/4885ALOX12 1699/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.