SCHEMBL16488408

SCHEMBL16488408

COc1ccc2cc(C(=O)C[C@H](C#N)c3cc(Cl)cc(Cl)c3)ccc2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.55
CYP1A2 P05177 2/20 0.49
ALDH1A1 P00352 1/20 0.49
HPGD P15428 1/20 0.49
CYP2C19 P33261 1/20 0.49
HSD17B10 Q99714 1/20 0.49
KDM4E B2RXH2 1/20 0.46
ABCB11 O95342 1/20 0.43
FFAR1 O14842 2/20 0.41
PTGS2 P35354 4/20 0.41
MGAM O43451 1/20 0.40
GAA P10253 1/20 0.40
SI P14410 1/20 0.40
MGAM2 Q2M2H8 1/20 0.40
KDM2B Q8NHM5 1/20 0.40
AKR1C3 P42330 5/20 0.40
AKR1C2 P52895 5/20 0.40
PTGS1 P23219 3/20 0.40
AKR1C1 Q04828 1/20 0.40
CDC42 P60953 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10309632 1.00 KMT2A (0.55) KMT2ACYP1A2ALDH1A1HPGDCYP2C19
SCHEMBL10309640 1.00 KMT2A (0.55) KMT2ACYP1A2ALDH1A1HPGDCYP2C19
SCHEMBL2662882 0.77 HSD17B10 (0.58) KMT2ACYP1A2ALDH1A1HPGDCYP2C19
SCHEMBL10309643 0.75 KMT2A (0.48) KMT2ACYP1A2ALDH1A1HPGDCYP2C19
SCHEMBL13385707 0.74 ALDH1A1 (0.50) KMT2ACYP1A2ALDH1A1HPGDCYP2C19
SCHEMBL8697184 0.74 TUBB4A (0.52) KMT2AALDH1A1KDM4EGAA
SCHEMBL1857883 0.74 CYP1A2 (0.61) KMT2ACYP1A2ALDH1A1HPGDCYP2C19
SCHEMBL13100658 0.74 KMT2A (0.79) KMT2AFFAR1
SCHEMBL8698087 0.73 L3MBTL1 (0.61) KMT2AALDH1A1MGAMGAASI
SCHEMBL23951761 0.73 KMT2A (0.39) KMT2ACYP1A2ALDH1A1HPGDCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2480077-B1 PYRROLIDINES AS GLUCAGON RECEPTOR ANTAGONISTS, COMPOSITIONS, AND METHODS FOR THEIR USE MERCK SHARP & DOHME (US) 2015-02-18 EP disclosed