SCHEMBL1648864

SCHEMBL1648864

COc1cccc(CNC(=O)c2cnc3cc(-c4cn[nH]c4)ccn23)c1

nearest known ligand 0.62

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 15/20 0.62
ROCK1 Q13464 9/20 0.62
PRKACA P17612 5/20 0.59
PRKACG P22612 5/20 0.59
PRKACB P22694 5/20 0.59
CLK1 P49759 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1648098 0.92 ROCK2 (0.55) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL1649817 0.88 ROCK2 (0.54) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL23384852 0.88 ROCK2 (0.50) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL1649577 0.87 CLK1 (0.75) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL1648756 0.87 AURKA (0.63) ROCK2ROCK1PRKACACLK1
SCHEMBL1649578 0.84 ROCK2 (0.61) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL19723671 0.84 CLK1 (0.61) ROCK2ROCK1PRKACACLK1
SCHEMBL1648234 0.83 ROCK2 (0.65) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL1649632 0.81 ROCK2 (0.61) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL1648102 0.81 CLK1 (0.52) ROCK2ROCK1PRKACAPRKACGPRKACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011050245-A1 BICYCLIC HETEROARYLS AS KINASE INHIBITORS FENG YANGBO (US) 2011-04-28 WO disclosed
WO-2011050245-A1 BICYCLIC HETEROARYLS AS KINASE INHIBITORS FENG YANGBO (US) 2011-04-28 WO disclosed