SCHEMBL16495337

SCHEMBL16495337

Nc1nc(N)c(Cc2ccc3[nH]ncc3c2)c(Cc2ccc3[nH]ncc3c2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
ROCK2 O75116 2/20 0.46
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
HPGD P15428 1/20 0.46
RAB9A P51151 1/20 0.46
KMT2A Q03164 1/20 0.46
ROCK1 Q13464 1/20 0.46
HIF1A Q16665 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
NOS1 P29475 3/20 0.43
MAPK1 P28482 2/20 0.40
QPCT Q16769 1/20 0.40
QPCTL Q9NXS2 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA2B P29275 1/20 0.40
ADORA1 P30542 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2598740 0.80 CYP17A1 (0.42) ALDH1A1ADORA3ADORA2AADORA2BADORA1
SCHEMBL2598585 0.77 CYP2A6 (0.45) ALDH1A1KDM4EMAPTHPGDTDP1
SCHEMBL16494934 0.75 DHFR (0.39) ALDH1A1KDM4EMAPTTDP1CYP2D6
SCHEMBL2598555 0.74 BACE1 (0.49) ALDH1A1CYP2D6ATMDHFR
SCHEMBL4230435 0.74 REN (0.50) ALDH1A1CYP2D6ATM
SCHEMBL16494607 0.74 ALDH1A1 (0.40) ALDH1A1CYP2D6ATMDHFR
SCHEMBL4218510 0.73 CYP2D6 (0.43) ALDH1A1MEN1KMT2ATDP1CYP2D6
SCHEMBL4218504 0.71 HSP90AB1 (0.53) ALDH1A1KDM4EMEN1HPGDKMT2A
SCHEMBL264211 0.71 ROCK2 (0.58) ALDH1A1ROCK2KDM4EMEN1GAA
SCHEMBL29728756 0.71 ROCK2 (0.58) ALDH1A1ROCK2KDM4EMEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2395001-A1 Novel pyrimidine derivatives Chemilia AB (SE) 2011-12-14 EP disclosed