SCHEMBL16498271

SCHEMBL16498271

c1ccc(-c2nc3cc(-c4ccc5[nH]c(-c6ccncc6)nc5c4)ccc3[nH]2)nc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.63
PKM P14618 4/20 0.63
RAB9A P51151 4/20 0.63
KDM4E B2RXH2 4/20 0.63
LMNA P02545 3/20 0.63
SMN1; SMN2 Q16637 3/20 0.63
MAPT P10636 2/20 0.63
KMT2A Q03164 1/20 0.63
METAP2 P50579 7/20 0.60
METAP1 P53582 6/20 0.60
HPGD P15428 3/20 0.60
MTOR P42345 1/20 0.60
ALDH1A1 P00352 2/20 0.57
PKN1 Q16512 1/20 0.57
PKN2 Q16513 1/20 0.57
CBFB Q13951 8/20 0.57
TP53 P04637 1/20 0.52
GAA P10253 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13866553 0.92 NPC1 (0.74) NPC1PKMRAB9AKDM4ELMNA
SCHEMBL16499527 0.88 NPC1 (0.55) NPC1PKMRAB9AKDM4ELMNA
SCHEMBL10351277 0.87 NPC1 (0.68) NPC1PKMRAB9AKDM4ELMNA
SCHEMBL16498963 0.87 NPC1 (0.54) NPC1PKMRAB9AKDM4ELMNA
SCHEMBL16497806 0.86 KDM4E (0.51) NPC1PKMRAB9AKDM4ELMNA
Ridinilazole SCHEMBL29379856 0.85 ALDH1A1 (0.66) NPC1PKMRAB9AKDM4ESMN1; SMN2
Ridinilazole SCHEMBL413723 0.85 ALDH1A1 (0.66) NPC1PKMRAB9AKDM4ESMN1; SMN2
SCHEMBL19994448 0.83 ALDH1A1 (0.59) NPC1PKMRAB9AKDM4ELMNA
SCHEMBL13866538 0.80 NPC1 (0.74) NPC1PKMRAB9AKDM4ELMNA
Ridinilazole SCHEMBL17867397 0.80 NPC1 (0.65) NPC1PKMRAB9AKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011151620-A1 COMPOUNDS FOR THE TREATMENT OF CLOSTRIDIUM DIFFICILE ASSOCIATED DISEASE SUMMIT CORPORATION PLC (GB) 2011-12-08 WO disclosed