SCHEMBL19994448

SCHEMBL19994448

c1cnc(-c2ccc3[nH]c(-c4ccncc4)nc3c2)nc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.59
KDM4E B2RXH2 4/20 0.59
PKN1 Q16512 4/20 0.59
PKN2 Q16513 4/20 0.59
HPGD P15428 3/20 0.55
HSD17B10 Q99714 2/20 0.55
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C9 P11712 1/20 0.55
CYP2C19 P33261 1/20 0.55
RHEB Q15382 1/20 0.55
NPC1 O15118 5/20 0.50
RAB9A P51151 4/20 0.50
GUSB P08236 1/20 0.48
SCD O00767 1/20 0.46
PDE10A Q9Y233 1/20 0.44
PDE4A P27815 1/20 0.44
PDE4B Q07343 1/20 0.44
PDE4C Q08493 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ridinilazole SCHEMBL413723 0.87 ALDH1A1 (0.66) ALDH1A1KDM4EPKN1PKN2HPGD
Ridinilazole SCHEMBL29379856 0.87 ALDH1A1 (0.66) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL19994736 0.83 AURKA (0.59) KDM4ENPC1RAB9AGUSBCHEK2
SCHEMBL16498271 0.83 NPC1 (0.63) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL30343733 0.83 AURKA (0.59) KDM4ENPC1RAB9AGUSBCHEK2
Ridinilazole SCHEMBL17867397 0.81 NPC1 (0.65) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL16498509 0.80 KDM4E (0.57) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL16499476 0.79 ALDH1A1 (0.65) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL22906080 0.79 ALDH1A1 (0.58) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL6263502 0.79 ALDH1A1 (0.58) ALDH1A1KDM4EPKN1PKN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12509465-B2 Benzoimidazole derivatives as anticancer agents CENTRE LEON BERARD (FR) 2025-12-30 US disclosed
EP-3515904-B1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2024-01-17 EP disclosed
EP-3515904-B1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2024-01-17 EP disclosed
CN-110234640-B Benzimidazole derivatives as anticancer agents 利昂贝拉尔中心 2023-04-07 CN disclosed
US-20220348587-A1 Benzoimidazole Derivatives As Anticancer Agents CENTRE LEON BERARD (FR) 2022-11-03 US disclosed
US-20220348587-A1 Benzoimidazole Derivatives As Anticancer Agents CENTRE LEON BERARD (FR) 2022-11-03 US disclosed
US-11384081-B2 Benzoimidazole derivatives as anticancer agents CENTRE LEON BERARD (FR) 2022-07-12 US disclosed
US-11384081-B2 Benzoimidazole derivatives as anticancer agents CENTRE LEON BERARD (FR) 2022-07-12 US disclosed
US-20210292328-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2021-09-23 US disclosed
US-20210292328-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2021-09-23 US disclosed
EP-3515904-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS Centre Leon Berard (FR) 2019-07-31 EP disclosed
WO-2018054989-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2018-03-29 WO disclosed
WO-2018054989-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2018-03-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12509465-B2 Benzoimidazole derivatives as anticancer agents CCAR2, MAPKAP1, BCOR ALDH1A1 3500/4885KDM4E 4285/4885PKN1 2537/4885
US-20210292328-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS TMBIM6, BAX, MAPK14 ALDH1A1 2866/4885KDM4E 1838/4885PKN1 796/4885
US-11384081-B2 Benzoimidazole derivatives as anticancer agents TMBIM6, BAX, MAPK14 ALDH1A1 2866/4885KDM4E 1838/4885PKN1 796/4885
US-20220348587-A1 Benzoimidazole Derivatives As Anticancer Agents TMBIM6, BAX, BCL2 ALDH1A1 2871/4885KDM4E 1858/4885PKN1 807/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.