Ridinilazole

Ridinilazole

SCHEMBL17867397

c1cc(-c2nc3cc(-c4ccc5nc(-c6ccncc6)[nH]c5c4)ccc3[nH]2)ccn1

nearest known ligand 0.65

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.65
RAB9A P51151 2/20 0.65
KDM4E B2RXH2 5/20 0.63
ALDH1A1 P00352 5/20 0.63
PKN1 Q16512 4/20 0.63
PKN2 Q16513 4/20 0.63
HPGD P15428 3/20 0.62
CYP3A4 P08684 2/20 0.62
HSD17B10 Q99714 2/20 0.62
CYP1A2 P05177 1/20 0.62
CYP2D6 P10635 1/20 0.62
CYP2C9 P11712 1/20 0.62
CYP2C19 P33261 1/20 0.62
RHEB Q15382 1/20 0.62
SCD O00767 1/20 0.58
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
RXFP1 Q9HBX9 2/20 0.54
CACNA1B Q00975 1/20 0.54
APBA1 Q02410 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ridinilazole SCHEMBL29785777 0.93 NPC1 (0.73) NPC1RAB9AKDM4EALDH1A1PKN1
Ridinilazole SCHEMBL19235713 0.93 NPC1 (0.73) NPC1RAB9AKDM4EALDH1A1PKN1
Ridinilazole SCHEMBL29613225 0.93 NPC1 (0.73) NPC1RAB9AKDM4EALDH1A1PKN1
Ridinilazole SCHEMBL413723 0.93 ALDH1A1 (0.66) NPC1RAB9AKDM4EALDH1A1PKN1
Ridinilazole SCHEMBL29379856 0.93 ALDH1A1 (0.66) NPC1RAB9AKDM4EALDH1A1PKN1
SCHEMBL14859469 0.88 NPC1 (0.52) NPC1RAB9AKDM4EALDH1A1PKN1
SCHEMBL14859468 0.88 NPC1 (0.52) NPC1RAB9AKDM4EALDH1A1PKN1
SCHEMBL14859401 0.88 NPC1 (0.52) NPC1RAB9AKDM4EALDH1A1PKN1
SCHEMBL16498433 0.87 ALDH1A1 (0.57) NPC1RAB9AKDM4EALDH1A1PKN1
SCHEMBL16497674 0.86 PKN1 (0.51) NPC1RAB9AKDM4EALDH1A1PKN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9763925-B2 Antibacterial compounds SUMMIT THERAPEUTICS PLC (GB) 2017-09-19 US claimed
US-20160184283-A1 ANTIBACTERIAL COMPOUNDS SUMMIT (OXFORD) LIMITED (GB) 2016-06-30 US claimed
US-20200290995-A1 Process for the Preparation of Crystalline Ridinilazole Using Acid Addition Salts SANDOZ AG (CH) 2020-09-17 US disclosed
WO-2019068383-A1 PROCESS FOR THE PREPARATION OF RIDINILAZOLE USING ACID ADDITION SALTS SANDOZ AG (CH) 2019-04-11 WO disclosed
US-9763925-B2 Antibacterial compounds SUMMIT THERAPEUTICS PLC (GB) 2017-09-19 US disclosed
US-20160184283-A1 ANTIBACTERIAL COMPOUNDS SUMMIT (OXFORD) LIMITED (GB) 2016-06-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160184283-A1 ANTIBACTERIAL COMPOUNDS MRPL21, RPN2, ALPI NPC1 512/4885RAB9A 1670/4885KDM4E 4769/4885
US-20200290995-A1 Process for the Preparation of Crystalline Ridinilazole Using Acid Addition Salts CYP3A5, CYP3A7, CYP3A4 NPC1 1676/4885RAB9A 1702/4885KDM4E 2756/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.