SCHEMBL1649998

SCHEMBL1649998

CC(C)(C)OC(=O)NCCCOc1c(C(=O)O)ccc(CS(=O)(=O)c2ccccc2)c1-c1ccoc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 10/20 0.41
CA2 P00918 10/20 0.41
CA12 O43570 5/20 0.41
CA9 Q16790 5/20 0.41
CYP1A1 P04798 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2B6 P20813 1/20 0.38
CYP2C19 P33261 1/20 0.38
CYP3A43 Q9HB55 1/20 0.38
POLB P06746 1/20 0.36
ALDH1A1 P00352 1/20 0.34
TP53 P04637 1/20 0.34
GLA P06280 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
XBP1 P17861 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HSD17B10 Q99714 1/20 0.34
IDO1 P14902 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1649052 0.86 CA1 (0.41) CA1CA2CA12CA9CYP1A1
SCHEMBL1648412 0.84 CA1 (0.40) CA1CA2CA12CA9CYP1A1
SCHEMBL1648181 0.83 CA1 (0.40) CA1CA2CA12CA9CYP1A1
Hydrochloric Acid SCHEMBL1648366 0.82 FABP4 (0.33) POLBFABP4FABP5
SCHEMBL1648648 0.81 ALDH1A1 (0.35) POLBALDH1A1METAP2FABP4FABP5
Hydrochloric Acid SCHEMBL14717753 0.80 ALDH1A1 (0.34) POLBALDH1A1METAP2FABP4FABP5
SCHEMBL1648204 0.79 CA12 (0.37) CA1CA2CA12CA9CYP1A1
SCHEMBL1649176 0.77 METAP2 (0.49) CA1CA2CA12CA9CYP1A1
SCHEMBL6844869 0.77 ALDH1A1 (0.40) CA1CA2CA12CA9CYP1A1
SCHEMBL1648514 0.75 MALT1 (0.42) CA1CA2CA12CA9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2486004-A2 SULPHONE COMPOUNDS AND METHODS OF MAKING AND USING SAME Zafgen Corporation (US) 2012-08-15 EP disclosed
WO-2011044506-A2 SULPHONE COMPOUNDS AND METHODS OF MAKING AND USING SAME ZAFGEN CORPORATION (US) 2011-04-14 WO disclosed