SCHEMBL1650229

SCHEMBL1650229

CCCCCCc1cc(Nc2ccccc2)ccc1N

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH3 Q9ULD8 1/20 0.42
TLR8 Q9NR97 3/20 0.41
MAPT P10636 7/20 0.41
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
KDM4E B2RXH2 2/20 0.41
GAA P10253 2/20 0.41
LMNA P02545 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
GFER P55789 1/20 0.41
ALDH1A1 P00352 7/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
MAPK1 P28482 2/20 0.41
CYP3A4 P08684 3/20 0.41
HTT P42858 2/20 0.41
ALOX12 P18054 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8680807 1.00 KCNH3 (0.42) KCNH3TLR8MAPTMEN1KMT2A
SCHEMBL6535929 0.94 MAPT (0.43) KCNH3TLR8MAPTMEN1KMT2A
SCHEMBL30392107 0.94 MAPT (0.43) KCNH3TLR8MAPTMEN1KMT2A
SCHEMBL536379 0.88 MAPT (0.46) MAPTMEN1KMT2AKDM4EGAA
SCHEMBL21278352 0.85 KCNH3 (0.44) KCNH3MAPTMEN1KMT2AGAA
N,N'-Diphenyl-P-Phenylenediamine SCHEMBL1415255 0.81 MAPT (0.48) KCNH3TLR8MAPTMEN1KMT2A
SCHEMBL2904304 0.81 ALDH1A1 (0.42) MAPTMEN1KMT2AKDM4EGAA
SCHEMBL3796679 0.81 MAPT (0.48) MAPTMEN1KMT2AKDM4EGAA
SCHEMBL10763021 0.80 PPARA (0.46) KCNH3MEN1KMT2APPARAPTGS2
SCHEMBL28175584 0.80 TLR8 (0.40) TLR8MAPTMEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 90 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3250620-A1 POLYURETHANE FOAMS BASED ON POLYETHER CARBONATE POLYOLS Covestro Deutschland AG (DE) 2017-12-06 EP disclosed
WO-2016120437-A1 POLYURETHANE FOAMS BASED ON POLYETHER CARBONATE POLYOLS COVESTRO DEUTSCHLAND AG (DE) 2016-08-04 WO disclosed
EP-2313421-A2 LIQUID OXYALKYLENE BRIDGED BIS- AND TRIS-PHOSPHITE ESTER MIXTURES BASF SE (DE) 2011-04-27 EP disclosed
WO-2010003809-A2 LIQUID OXYALKYLENE BRIDGED BIS- AND TRIS-PHOSPHITE ESTER MIXTURES BASF SE (DE) 2010-01-14 WO disclosed
EP-2125945-A1 PROCESSING STABILIZERS FOR RUBBER COMPOUNDING BASF SE (DE) 2009-12-02 EP disclosed
EP-2122020-A1 WETTABLE POLYESTER FIBERS AND FABRICS Ciba Holding Inc. (CH) 2009-11-25 EP disclosed
WO-2008113702-A1 PROCESSING STABILIZERS FOR RUBBER COMPOUNDING BASF SE (CH) 2008-09-25 WO disclosed
EP-1951938-A2 WETTABLE POLYESTER FIBERS AND FABRICS Ciba Holding Inc. (CH) 2008-08-06 EP disclosed
WO-2008090060-A1 WETTABLE POLYESTER FIBERS AND FABRICS CIBA HOLDING INC. (CH) 2008-07-31 WO disclosed
EP-1943236-A2 PROCESS FOR THE SYNTHESIS OF AMINE ETHERS Ciba Holding Inc. (CH) 2008-07-16 EP disclosed
WO-1998054175-A1 BLOCK OLIGOMERS CONTAINING 1-HYDROCARBYLOXY-2,2,6,6-TETRAMETHYL-4-PIPERIDYL GROUPS AS STABILIZERS FOR ORGANIC MATERIALS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 1998-12-03 WO disclosed
WO-1998054174-A1 BLOCK OLIGOMERS CONTAINING 1-HYDROCARBYLOXY-2,2,6,6-TETRAMETHYL-4-PIPERIDYL GROUPS AS STABILIZERS FOR ORGANIC MATERIALS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 1998-12-03 WO disclosed
EP-0880557-A1 STABILISATION OF POLYOLEFIN-RECYCLATES Ciba SC Holding AG (CH) 1998-12-02 EP disclosed
WO-1998046342-A2 PREPARATION OF LOW-DUST STABILISERS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 1998-10-22 WO disclosed
EP-0858449-A1 THERMALLY STABLE HINDERED AMINES AS STABILIZERS Ciba SC Holding AG (CH) 1998-08-19 EP disclosed
WO-1998028361-A1 LIGHT-STABILISED FLAMEPROOF STYRENE HOMOPOLYMERS AND COPOLYMERS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 1998-07-02 WO disclosed
WO-1998003489-A1 POLYOXYALKENE SUBSTITUTED AND BRIDGED TRIAZINE, BENZOTRIAZOLE AND BENZOPHENONE DERIVATIVES AS UV ABSORBERS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 1998-01-29 WO disclosed
WO-1997036880-A1 AMINO- AND HYDROXYSUBSTITUTED TRIPHENYL-S-TRIAZINES AS STABILIZERS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 1997-10-09 WO disclosed
WO-1997030112-A1 STABILISATION OF POLYOLEFIN-RECYCLATES CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 1997-08-21 WO disclosed
WO-1997013752-A1 THERMALLY STABLE HINDERED AMINES AS STABILIZERS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 1997-04-17 WO disclosed