SCHEMBL16503582

SCHEMBL16503582

CC=C(O)c1ccc2cccc(-c3cc(Cl)ccc3F)c2c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MEN1 O00255 1/20 0.34
RAB9A P51151 1/20 0.34
KMT2A Q03164 1/20 0.34
AKR1C3 P42330 1/20 0.34
AKR1C2 P52895 1/20 0.34
SERPINE1 P05121 1/20 0.32
TRPV1 Q8NER1 2/20 0.32
PLA2G2D Q9UNK4 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
CHRM5 P08912 1/20 0.32
CHRM1 P11229 1/20 0.32
CHRM3 P20309 1/20 0.32
MAPT P10636 1/20 0.32
APEX1 P27695 1/20 0.32
GRM2 Q14416 1/20 0.31
CYP2A6 P11509 1/20 0.31
HSD11B1 P28845 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7919880 0.84 PLA2G2D (0.48) MEN1RAB9AKMT2ASERPINE1TRPV1
SCHEMBL16503581 0.83 AKR1C3 (0.36) MEN1RAB9AKMT2AAKR1C3AKR1C2
SCHEMBL16503577 0.80 ESR1 (0.34) LMNAMEN1KMT2ATRPV1MAPT
SCHEMBL7911019 0.80 PLAU (0.47) MEN1RAB9AKMT2AMAPTPLAU
SCHEMBL7923148 0.75 HTR5A (0.50)
SCHEMBL16502526 0.75 GRM2 (0.47) MEN1RAB9AKMT2AAKR1C3AKR1C2
SCHEMBL16503575 0.73 GABRG2 (0.35) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL16503550 0.73 KDM4E (0.36) SMN1; SMN2MEN1RAB9AKMT2AF2
SCHEMBL16503496 0.72 HTR2C (0.43) LMNASMN1; SMN2RAB9AMAPTF2
SCHEMBL7918358 0.71 TRPV1 (0.46) RAB9ASERPINE1TRPV1PLA2G2D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2394987-A1 ACYLGUANIDINE DERIVATIVE Astellas Pharma Inc. (JP) 2011-12-14 EP disclosed