SCHEMBL16503577

SCHEMBL16503577

CC=C(O)c1ccc2cccc(-c3c(F)ccc(O)c3Cl)c2c1

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 7/20 0.34
ESR2 Q92731 7/20 0.34
HSD17B14 Q9BPX1 1/20 0.32
THRA P10827 1/20 0.31
THRB P10828 1/20 0.31
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
HTT P42858 1/20 0.31
KMT2A Q03164 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
TRPV1 Q8NER1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7915371 0.85 PLA2G2D (0.44) ESR1ESR2HSD17B14THRBMEN1
SCHEMBL16502604 0.81 LCK (0.45) MEN1ALDH1A1LMNAMAPTHTT
SCHEMBL16503582 0.80 LMNA (0.34) MEN1LMNAMAPTKMT2ATRPV1
SCHEMBL7918251 0.77 HTR5A (0.50)
SCHEMBL16503581 0.77 AKR1C3 (0.36) MEN1ALDH1A1MAPTKMT2ACYP1A2
SCHEMBL7915369 0.73 PLA2G2D (0.46) HSD17B14THRBMEN1ALDH1A1LMNA
SCHEMBL16503571 0.71 MCL1 (0.35) MEN1ALDH1A1MAPTHTTKMT2A
SCHEMBL16502500 0.70 PLA2G2D (0.49) MEN1KMT2ATRPV1
SCHEMBL7921825 0.70 PLA2G2D (0.46) HSD17B14THRBMEN1ALDH1A1LMNA
SCHEMBL16503575 0.70 GABRG2 (0.35) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2394987-A1 ACYLGUANIDINE DERIVATIVE Astellas Pharma Inc. (JP) 2011-12-14 EP disclosed